SCHEMBL28031645

SCHEMBL28031645

O=C(O)c1nccnc1Oc1cccc(Br)c1

nearest known ligand 0.46

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
EGFR P00533 3/20 0.46
MRGPRX4 Q96LA9 1/20 0.45
ABCG2 Q9UNQ0 1/20 0.43
KDM4E B2RXH2 6/20 0.42
ALDH1A1 P00352 6/20 0.42
KMT2A Q03164 3/20 0.42
CYP1A2 P05177 2/20 0.42
LMNA P02545 1/20 0.42
CYP2C9 P11712 1/20 0.42
TSHR P16473 1/20 0.42
CYP2C19 P33261 1/20 0.42
KDR P35968 1/20 0.41
MAPT P10636 2/20 0.40
GAA P10253 1/20 0.40
RECQL P46063 1/20 0.40
MAOB P27338 1/20 0.40
HSD17B10 Q99714 1/20 0.39
SMN1; SMN2 Q16637 1/20 0.39
MCL1 Q07820 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28030562 0.82 HAO1 (0.45) KDM4EKMT2ACYP1A2CYP2C19
SCHEMBL10970875 0.81 TDP1 (0.52) EGFRALDH1A1KMT2ACYP1A2CYP2C9
SCHEMBL19977428 0.75 EGFR (0.50) EGFRABCG2ALDH1A1KMT2ACYP1A2
SCHEMBL6136728 0.74 EGFR (0.52) EGFRABCG2ALDH1A1KMT2ACYP1A2
SCHEMBL28035897 0.72 KMT2A (0.47) KDM4EKMT2ACYP1A2CYP2C9CYP2C19
SCHEMBL20704068 0.72 MRGPRX4 (0.44) EGFRMRGPRX4ABCG2ALDH1A1KMT2A
SCHEMBL23319939 0.71 HAO1 (0.41) MRGPRX4KDM4EKMT2ACYP1A2MAPT
SCHEMBL26195027 0.71 ICAM1 (0.41) EGFRMRGPRX4KDM4EALDH1A1KMT2A
SCHEMBL8476094 0.70 ALDH1A1 (0.51) KDM4EALDH1A1KMT2A
SCHEMBL5519221 0.70 SRD5A2 (0.61) MRGPRX4KDM4ECYP1A2CYP2C9CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105017166-A Preparation method of 3-(3-bromine phenoxy) pyrazine-2-carboxylic acid CHANGSHA SHENCHENG BIOLOG TECHNOLOGY CO LTD 2015-11-04 CN disclosed
CN-105017166-A Preparation method of 3-(3-bromine phenoxy) pyrazine-2-carboxylic acid CHANGSHA SHENCHENG BIOLOG TECHNOLOGY CO LTD 2015-11-04 CN disclosed