SCHEMBL28031940

SCHEMBL28031940

Cc1cccc2c(O)nc(-c3cccnc3)nc12

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 4/20 0.55
HTT P42858 3/20 0.55
LMNA P02545 3/20 0.55
CYP2A6 P11509 4/20 0.46
ADORA3 P0DMS8 1/20 0.45
TSHR P16473 4/20 0.44
CYP3A4 P08684 4/20 0.44
SMN1; SMN2 Q16637 4/20 0.44
ALDH1A1 P00352 4/20 0.44
CYP2D6 P10635 3/20 0.44
CYP2C9 P11712 3/20 0.44
CYP1A2 P05177 3/20 0.44
CLK4 Q9HAZ1 3/20 0.44
HPGD P15428 3/20 0.44
HSD17B10 Q99714 2/20 0.44
CYP2C19 P33261 2/20 0.44
RAB9A P51151 2/20 0.44
MEN1 O00255 1/20 0.44
GLA P06280 1/20 0.44
KMT2A Q03164 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2155051 0.81 SMN1; SMN2 (0.44) KDM4EHTTLMNACYP2A6TSHR
SCHEMBL2215084 0.78 NPC1 (0.52) KDM4ELMNAADORA3TSHRCYP3A4
SCHEMBL14358640 0.74 CYP11B1 (0.43) KDM4EHTTLMNACYP2A6TSHR
SCHEMBL16183770 0.74 S1PR1 (0.45) KDM4ELMNATSHRSMN1; SMN2ALDH1A1
SCHEMBL14474797 0.72 MAPT (0.52) KDM4EHTTLMNAADORA3CYP3A4
SCHEMBL14727925 0.72 KMT2A (0.51) KDM4EHTTLMNATSHRCYP3A4
SCHEMBL12339131 0.72 CYP2A6 (0.54) KDM4EHTTLMNACYP2A6TSHR
SCHEMBL31620698 0.71 KDM4E (1.00) KDM4EHTTLMNATSHRSMN1; SMN2
SCHEMBL2155114 0.71 CHRNB2 (0.43) KDM4EHTTLMNACYP2A6TSHR
SCHEMBL9133519 0.71 TDO2 (0.50) KDM4EHTTLMNATSHRCYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105218516-A Therapeutic compounds and related methods of use OTSUKA PHARMA CO LTD 2016-01-06 CN disclosed
CN-102883723-B Therapeutic compounds and related methods of use OTSUKA PHARMACEUTICAL CO.,LTD. (JP) 2015-09-16 CN disclosed