SCHEMBL28032410

SCHEMBL28032410

O=C(c1cccc2ncc3ccccc3c12)c1cccc2ncc3ccccc3c12

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 1/20 0.52
GPR3 P46089 1/20 0.52
CDC25B P30305 2/20 0.45
NR4A1 P22736 1/20 0.42
NR4A2 P43354 1/20 0.42
NR4A3 Q92570 1/20 0.42
MGAM O43451 1/20 0.40
PIM1 P11309 1/20 0.40
CNR2 P34972 3/20 0.40
TOP2A P11388 1/20 0.39
TOP2B Q02880 1/20 0.39
ALDH1A1 P00352 2/20 0.39
MMP3 P08254 1/20 0.39
HDAC8 Q9BY41 1/20 0.39
HPGD P15428 1/20 0.39
ALOX15 P16050 1/20 0.39
HSD17B10 Q99714 1/20 0.39
MEN1 O00255 2/20 0.38
KMT2A Q03164 2/20 0.38
MAPT P10636 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18663455 0.91 KDM4E (0.46) KDM4EGPR3CDC25BNR4A1NR4A2
SCHEMBL5358558 0.89 KDM4E (0.50) KDM4EGPR3CDC25BNR4A1NR4A2
SCHEMBL5358564 0.89 NR4A1 (0.53) KDM4EGPR3CDC25BNR4A1NR4A2
SCHEMBL8230482 0.87 PIM1 (0.50) KDM4EGPR3PIM1ALDH1A1MEN1
SCHEMBL3862098 0.87 LIG1 (0.46) KDM4EGPR3MGAMALDH1A1HPGD
SCHEMBL27546968 0.84 KDM4E (0.46) KDM4EGPR3NR4A1NR4A2NR4A3
SCHEMBL27656146 0.82 KDM4E (0.44) KDM4EGPR3CDC25BNR4A1NR4A2
SCHEMBL27656141 0.82 KDM4E (0.44) KDM4EGPR3CDC25BNR4A1NR4A2
SCHEMBL30075099 0.82 KDM4E (0.50) KDM4EGPR3CDC25BNR4A1NR4A2
SCHEMBL29598792 0.77 KDM4E (0.57) KDM4EGPR3ALDH1A1HDAC8HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 16 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-116854635-A Synthesis method of phenanthridine-6 (5H) -ketone compound 安徽中烟工业有限责任公司 2023-10-10 CN disclosed
CN-116854635-A Synthesis method of phenanthridine-6 (5H) -ketone compound 安徽中烟工业有限责任公司 2023-10-10 CN disclosed
CN-108191834-B Preparation method of benzo-fused N-heterocyclic compound 中山大学 2020-10-16 CN disclosed
CN-110698430-A Thiaphenanthrone derivative, method for synthesizing the same, and electronic device containing the same 苏州久显新材料有限公司 2020-01-17 CN disclosed
CN-110698430-A Thiaphenanthrone derivative, method for synthesizing the same, and electronic device containing the same 苏州久显新材料有限公司 2020-01-17 CN disclosed
CN-110256346-A Phenanthridines ketone compounds and preparation method and application with BRD4 albumen inhibiting effect 浙江省医学科学院 2019-09-20 CN disclosed
CN-110256346-A Phenanthridines ketone compounds and preparation method and application with BRD4 albumen inhibiting effect 浙江省医学科学院 2019-09-20 CN disclosed
CN-109320497-A A method of phenanthridines ketone compounds are prepared by copper compound induction 广州大学 2019-02-12 CN disclosed
CN-108948029-A Phenanthridinone derivative, and synthesis method and anti-tumor application thereof 华中科技大学 2018-12-07 CN disclosed
CN-108948029-A Phenanthridinone derivative, and synthesis method and anti-tumor application thereof 华中科技大学 2018-12-07 CN disclosed
CN-108191834-A A kind of preparation method of benzo-fused N- heterocyclic compounds 中山大学 2018-06-22 CN disclosed
CN-104926723-B Synthetic method of phenanthridine ketone compounds 洛阳师范学院 2017-04-19 CN disclosed
CN-104926723-B Synthetic method of phenanthridine ketone compounds 洛阳师范学院 2017-04-19 CN disclosed
CN-104926723-B Synthetic method of phenanthridine ketone compounds 洛阳师范学院 2017-04-19 CN disclosed
CN-104926723-A Synthetic method of phenanthridine ketone compounds UNIV LUOYANG NORMAL 2015-09-23 CN disclosed
CN-104926723-A Synthetic method of phenanthridine ketone compounds UNIV LUOYANG NORMAL 2015-09-23 CN disclosed