SCHEMBL2803344

SCHEMBL2803344

NS(=O)(=O)c1ccccc1S(=O)(=O)NC(=O)c1ccc(Br)c(OCC2CC2)c1

nearest known ligand 0.55

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
PTGES O14684 2/20 0.55
PDE4B Q07343 7/20 0.43
PDE4A P27815 6/20 0.43
PDE4C Q08493 6/20 0.43
PDE4D Q08499 6/20 0.43
P2RX4 Q99571 4/20 0.42
KAT6A Q92794 4/20 0.41
CYSLTR2 Q9NS75 1/20 0.40
CYSLTR1 Q9Y271 1/20 0.40
BCL2L1 Q07817 1/20 0.38
MCL1 Q07820 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13066257 0.86 PTGES (0.54) PTGESPDE4BPDE4APDE4CPDE4D
SCHEMBL2803916 0.85 PTGES (0.51) PTGESPDE4BPDE4APDE4CPDE4D
SCHEMBL2802046 0.83 PTGES (0.62) PTGESPDE4BPDE4APDE4CPDE4D
SCHEMBL2803278 0.82 PTGES (0.61) PTGESPDE4BPDE4APDE4CPDE4D
SCHEMBL2802679 0.82 PTGES (0.48) PTGESKAT6ACYSLTR2CYSLTR1
SCHEMBL2802184 0.82 PTGES (0.51) PTGESKAT6A
SCHEMBL2805238 0.82 PTGES (0.48) PTGES
SCHEMBL2802125 0.82 PTGES (0.51) PTGESKAT6ACYSLTR2CYSLTR1
SCHEMBL978258 0.81 PTGES (0.52) PTGESCYSLTR2CYSLTR1
SCHEMBL978260 0.81 PTGES (0.64) PTGESCYSLTR2CYSLTR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010132016-A1 BIS-(SULFONYLAMINO) DERIVATIVES FOR TREATMENT OF PAIN AND INFLAMMATION ASTRAZENECA AB (SE) 2010-11-18 WO disclosed
US-20100292279-A1 Bis-(Sulfonylamino) Derivatives in Therapy ASTRAZENECA AB (SE) 2010-11-18 US disclosed
US-20100292279-A1 Bis-(Sulfonylamino) Derivatives in Therapy ASTRAZENECA AB (SE) 2010-11-18 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20100292279-A1 Bis-(Sulfonylamino) Derivatives in Therapy PTGER1, SULT2A1, SULT1E1 PTGES 9/4885PDE4B 1521/4885PDE4A 1098/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.