SCHEMBL28033926

SCHEMBL28033926

Oc1cccc2ccc(CNCc3ccccc3)nc12

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PKM P14618 1/20 0.49
HDAC1 Q13547 4/20 0.46
HDAC2 Q92769 3/20 0.46
HDAC8 Q9BY41 2/20 0.46
HDAC6 Q9UBN7 2/20 0.46
CYP1A2 P05177 2/20 0.45
HIF1A Q16665 2/20 0.45
ALOX15 P16050 2/20 0.45
CYP2D6 P10635 1/20 0.45
KMT2A Q03164 3/20 0.44
LMNA P02545 2/20 0.44
TDP1 Q9NUW8 2/20 0.44
MAPT P10636 1/20 0.44
KDM4E B2RXH2 2/20 0.44
METAP2 P50579 1/20 0.44
PLAU P00749 1/20 0.44
NCF1 P14598 1/20 0.44
MPO P05164 2/20 0.43
POLB P06746 1/20 0.43
ALOX12 P18054 2/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9471806 0.84 METAP2 (0.49) HDAC1HDAC2HDAC8HDAC6CYP1A2
SCHEMBL8344444 0.82 KDM4E (0.52) HDAC8CYP1A2HIF1AALOX15KMT2A
SCHEMBL19622955 0.81 CA12 (0.46) HDAC8CYP1A2HIF1AALOX15KMT2A
SCHEMBL360767 0.81 KMT2A (0.49) CYP1A2HIF1AKMT2ALMNATDP1
SCHEMBL7562315 0.81 KMT2A (0.50) HDAC1HDAC2HDAC8HDAC6CYP1A2
SCHEMBL7133311 0.80 KCNH2 (0.56) HDAC8CYP1A2HIF1AKMT2ALMNA
Hydrochloric Acid SCHEMBL6053093 0.80 KMT2A (0.47) CYP1A2HIF1AKMT2ALMNATDP1
SCHEMBL12593364 0.78 METAP2 (0.49) HDAC8CYP1A2HIF1AALOX15KMT2A
SCHEMBL4040914 0.77 KMT2A (0.45) HDAC8HDAC6CYP1A2HIF1ACYP2D6
SCHEMBL31238931 0.76 MEN1 (0.54) PKMHDAC1KMT2ATDP1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-104994853-A Dihydro-6-azaphenalene derivatives for the treatment of cns, oncological diseases and related disorders WARNER BABCOCK INST FOR GREEN CHEMISTRY LLC 2015-10-21 CN disclosed