SCHEMBL280340

SCHEMBL280340

CCNC1CCN(CC(=O)c2ccc(C)s2)C1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 2/20 0.40
RAB9A P51151 2/20 0.40
CCR2 P41597 2/20 0.39
ALDH1A1 P00352 3/20 0.39
TAS1R3 Q7RTX0 1/20 0.39
TAS1R1 Q7RTX1 1/20 0.39
ADORA2A P29274 2/20 0.38
ADORA1 P30542 2/20 0.38
KCNH2 Q12809 1/20 0.38
MEN1 O00255 1/20 0.38
KMT2A Q03164 1/20 0.38
LMNA P02545 1/20 0.38
POLB P06746 1/20 0.38
RECQL P46063 1/20 0.38
L3MBTL1 Q9Y468 1/20 0.38
HPGD P15428 1/20 0.38
ACKR3 P25106 2/20 0.37
HTR1A P08908 1/20 0.36
USP28 Q96RU2 1/20 0.36
USP25 Q9UHP3 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL279886 0.80 ALDH1A1 (0.42) NPC1RAB9AALDH1A1TAS1R3TAS1R1
SCHEMBL279992 0.74 DAO (0.44) NPC1RAB9AALDH1A1TAS1R3TAS1R1
SCHEMBL279616 0.73 RAB9A (0.49) NPC1RAB9AALDH1A1MEN1KMT2A
SCHEMBL279637 0.72 ALDH1A1 (0.49) NPC1RAB9AALDH1A1MEN1KMT2A
SCHEMBL279862 0.71 ALDH1A1 (0.51) RAB9AALDH1A1MEN1KMT2ALMNA
SCHEMBL279970 0.71 DAO (0.43) NPC1RAB9AALDH1A1MEN1KMT2A
SCHEMBL18419027 0.70 KMT2A (0.47) CCR2ALDH1A1MEN1KMT2ALMNA
SCHEMBL279617 0.70 DAO (0.42) NPC1RAB9AALDH1A1MEN1KMT2A
SCHEMBL660676 0.69 KMT2A (0.38) RAB9AALDH1A1MEN1KMT2ALMNA
SCHEMBL28853888 0.69 ADORA2A (0.36) CCR2ADORA2AADORA1KCNH2MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8134013-B2 Amide compound and thrombopoietin receptor activator NISSAN CHEMICAL INDUSTRIES, LTD. (JP) 2012-03-13 US disclosed
US-20090131659-A1 AMIDE COMPOUND AND THROMBOPOIETIN RECEPTOR ACTIVATOR NISSAN CHEMICAL INDUSTRIES, LTD. (JP) 2009-05-21 US disclosed
EP-1845090-A1 AMIDE COMPOUND AND THROMBOPOIETIN RECEPTOR ACTIVATOR Nissan Chemical Industries, Ltd. (JP) 2007-10-17 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20090131659-A1 AMIDE COMPOUND AND THROMBOPOIETIN RECEPTOR ACTIVATOR TEK, PTAFR, MPL NPC1 3107/4885RAB9A 2458/4885CCR2 622/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.