SCHEMBL28034152

SCHEMBL28034152

N#CN(Cc1cccnc1)Cc1cc(C(F)(F)F)cc(C(F)(F)F)c1

nearest known ligand 0.43

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
CHRNB2 P17787 2/20 0.43
CHRNA4 P43681 2/20 0.43
NR1H3 Q13133 3/20 0.43
NR1D1 P20393 2/20 0.43
ALDH1A1 P00352 1/20 0.42
CACNA1H O95180 1/20 0.41
GPBAR1 Q8TDU6 6/20 0.40
NR1H2 P55055 1/20 0.40
TACR1 P25103 2/20 0.39
HIF1A Q16665 1/20 0.39
EPAS1 Q99814 1/20 0.39
KDM4E B2RXH2 1/20 0.39
POLB P06746 1/20 0.39
CYP3A4 P08684 1/20 0.39
CYP3A5 P20815 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28822559 0.81 NR1H3 (0.47) CHRNB2CHRNA4NR1H3NR1D1ALDH1A1
SCHEMBL7382021 0.73 CACNA1H (0.45) CACNA1HGPBAR1HIF1AKDM4EPOLB
SCHEMBL1600409 0.72 TACR1 (0.38) ALDH1A1TACR1CYP3A4
SCHEMBL1601025 0.72 SLC6A4 (0.40) ALDH1A1TACR1
SCHEMBL25797239 0.70 CYP3A4 (0.53) CHRNB2CHRNA4NR1H3NR1D1GPBAR1
SCHEMBL7381239 0.70 CACNA1H (0.45) CACNA1HHIF1AKDM4EPOLBCYP3A4
SCHEMBL27602785 0.69 HIF1A (0.65) CHRNB2CHRNA4NR1H3ALDH1A1NR1H2
SCHEMBL30062626 0.69 CACNA1H (0.53) NR1H3NR1D1CACNA1HKDM4EPOLB
SCHEMBL16606309 0.68 CHRNB2 (0.58) CHRNB2CHRNA4ALDH1A1KDM4E
SCHEMBL19687731 0.68 NR1H3 (0.41) CHRNB2CHRNA4NR1H3NR1D1CACNA1H

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-103102303-B As the benzyl amine derivative of CETP inhibitor DR. REDDY'S LABORATORIES LTD. (IN) 2015-10-28 CN disclosed