SCHEMBL25797239

SCHEMBL25797239

CC(=O)N(Cc1cccnc1)c1cc(C(F)(F)F)cc(C(F)(F)F)c1

nearest known ligand 0.53

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 2/20 0.53
L3MBTL1 Q9Y468 1/20 0.49
HDAC6 Q9UBN7 1/20 0.48
TP53 P04637 3/20 0.47
GPBAR1 Q8TDU6 1/20 0.47
HIF1A Q16665 1/20 0.47
EPAS1 Q99814 1/20 0.47
TSPO P30536 1/20 0.46
SORT1 Q99523 1/20 0.46
NR1H3 Q13133 2/20 0.46
NR1H2 P55055 1/20 0.46
RIPK1 Q13546 1/20 0.44
PDK1 Q15118 1/20 0.44
CHRNB2 P17787 1/20 0.43
CHRNA4 P43681 1/20 0.43
NR1D1 P20393 1/20 0.43
LMNA P02545 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18763043 0.84 GSTO1 (0.50) CYP3A4HIF1AEPAS1SORT1NR1H3
SCHEMBL10985162 0.79 CYP3A4 (0.67) CYP3A4L3MBTL1TP53PDK1CHRNB2
SCHEMBL10992280 0.76 CYP3A4 (0.60) CYP3A4L3MBTL1TP53PDK1CHRNB2
SCHEMBL21168598 0.75 CYP3A4 (0.46) CYP3A4L3MBTL1TP53TSPOPDK1
SCHEMBL6733814 0.72 GRM2 (0.62) CYP3A4L3MBTL1TP53TSPOLMNA
SCHEMBL19687731 0.72 NR1H3 (0.41) HIF1AEPAS1SORT1NR1H3NR1H2
SCHEMBL2187051 0.72 KDM4E (0.61) CYP3A4RIPK1CHRNB2CHRNA4LMNA
SCHEMBL10560010 0.71 GRM2 (0.57) CYP3A4HDAC6
SCHEMBL7748094 0.71 TBXAS1 (0.62) CYP3A4L3MBTL1HDAC6TP53
SCHEMBL7748091 0.71 TBXAS1 (0.62) CYP3A4L3MBTL1HDAC6TP53

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023125751-A1 DIA-BASED QUANTITATIVE CHEMICAL PROTEOMICS TARGET SCREENING METHOD 北京大学 2023-07-06 WO disclosed