SCHEMBL28035287

SCHEMBL28035287

Oc1cc2cccc(O)c2cn1

nearest known ligand 0.61

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
IDO1 P14902 1/20 0.61
TDO2 P48775 1/20 0.61
MAPT P10636 1/20 0.48
KDM4E B2RXH2 5/20 0.47
PLAU P00749 1/20 0.47
MAPKAPK2 P49137 1/20 0.47
CYP1A2 P05177 1/20 0.46
HSD17B1 P14061 5/20 0.44
HSD17B2 P37059 5/20 0.44
ESR1 P03372 2/20 0.44
ESR2 Q92731 2/20 0.44
GRIN2D O15399 1/20 0.43
GRIN2A Q12879 1/20 0.43
GRIN2B Q13224 1/20 0.43
GRIN2C Q14957 1/20 0.43
CTDSP1 Q9GZU7 1/20 0.42
MMP2 P08253 1/20 0.41
CHRM1 P11229 1/20 0.41
TSHR P16473 1/20 0.41
COMT P21964 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2749558 0.80 CYP1A2 (0.47) IDO1TDO2KDM4ECYP1A2HSD17B1
SCHEMBL1564051 0.80 IDO1 (0.57) IDO1TDO2MAPTKDM4EPLAU
SCHEMBL1397048 0.80 IDO1 (0.41) IDO1TDO2MAPTKDM4EHSD17B1
SCHEMBL2747921 0.80 IDO1 (0.41) IDO1TDO2MAPTKDM4EPLAU
SCHEMBL2748752 0.80 CHEK1 (0.46) IDO1TDO2MAPTKDM4ECYP1A2
SCHEMBL12611446 0.79 IDO1 (0.47) IDO1TDO2MAPTKDM4EHSD17B1
SCHEMBL8341742 0.78 ALDH1A1 (0.52) IDO1TDO2MAPTKDM4ECYP1A2
SCHEMBL2749000 0.76 HSD17B1 (0.43) IDO1TDO2MAPTKDM4EHSD17B1
SCHEMBL1397032 0.76 MAPT (0.49) IDO1TDO2MAPTKDM4EALDH1A1
SCHEMBL2749751 0.76 HTT (0.49) IDO1TDO2MAPTKDM4EESR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105399669-B A kind of dihydroxy isoquinolin and its methods and applications prepared from centipede 中国药科大学 2019-05-03 CN claimed
CN-105399669-A Dihydroxy isoquinoline and preparation method and application thereof from centipedes UNIV CHINA PHARMA 2016-03-16 CN claimed
CN-105399669-B A kind of dihydroxy isoquinolin and its methods and applications prepared from centipede 中国药科大学 2019-05-03 CN disclosed
CN-105399669-B A kind of dihydroxy isoquinolin and its methods and applications prepared from centipede 中国药科大学 2019-05-03 CN disclosed
CN-105004809-B Centipede medicinal material quality detection method 鲁南制药集团股份有限公司 2017-02-08 CN disclosed
CN-105399669-A Dihydroxy isoquinoline and preparation method and application thereof from centipedes UNIV CHINA PHARMA 2016-03-16 CN disclosed
CN-105399669-A Dihydroxy isoquinoline and preparation method and application thereof from centipedes UNIV CHINA PHARMA 2016-03-16 CN disclosed
CN-105004809-A Centipede medicinal material quality control method LUNAN PHARM GROUP CORP 2015-10-28 CN disclosed