SCHEMBL28035946

SCHEMBL28035946

O=C1Nc2ccc(-c3ccc(F)cc3)cc2C1O

nearest known ligand 0.44

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
PGR P06401 8/20 0.44
ERCC1 P07992 1/20 0.38
ERCC4 Q92889 1/20 0.38
MAPT P10636 2/20 0.38
HDAC1 Q13547 1/20 0.37
HDAC6 Q9UBN7 1/20 0.37
HTR7 P34969 1/20 0.36
TNKS2 Q9H2K2 1/20 0.36
NTRK1 P04629 1/20 0.34
BCL2L1 Q07817 1/20 0.34
BAD Q92934 1/20 0.34
PDK2 Q15119 1/20 0.34
PTGDR Q13258 1/20 0.34
PTGDR2 Q9Y5Y4 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11211006 0.83 PDE3B (0.49) PGR
SCHEMBL10714214 0.77 PGR (0.42) PGRMAPTHDAC1HDAC6HTR7
SCHEMBL8210790 0.73 MEN1 (0.39) PGRMAPT
SCHEMBL14438188 0.73 NQO2 (0.50) MAPT
SCHEMBL3423085 0.70 CA1 (0.41)
SCHEMBL17260218 0.69 GSK3B (0.49) MAPT
SCHEMBL2056415 0.69 MAPT (0.42) PGRMAPT
SCHEMBL2054640 0.69 MEN1 (0.42) PGRMAPT
SCHEMBL2056355 0.69 SMN1; SMN2 (0.42) PGRMAPT
SCHEMBL20600322 0.67 IDO1 (0.50) MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105102452-B The ketones derivant of 5 (base of 3,5 dimethyl isoxazole 4) indoline 2 of substitution 百济神州有限公司 2018-01-26 CN disclosed
CN-105102452-A Substituted5-(3,5-dimethylisoxazol-4-yl)indoline-2-ones BEIGENE LTD 2015-11-25 CN disclosed