SCHEMBL28036654

SCHEMBL28036654

COc1ccc(C(COC=O)c2scnc2C)cc1

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SLC6A3 Q01959 6/20 0.36
SLC6A4 P31645 1/20 0.36
CYP17A1 P05093 1/20 0.35
BACE1 P56817 1/20 0.34
FFAR1 O14842 3/20 0.32
CYP19A1 P11511 1/20 0.32
KDM4E B2RXH2 2/20 0.32
PKM P14618 1/20 0.32
LMNA P02545 2/20 0.32
HTT P42858 2/20 0.32
MITF O75030 1/20 0.32
CNR1 P21554 1/20 0.32
CNR2 P34972 1/20 0.32
GPR35 Q9HC97 1/20 0.32
GPR55 Q9Y2T6 1/20 0.32
XBP1 P17861 1/20 0.32
MAPK1 P28482 1/20 0.32
NPSR1 Q6W5P4 1/20 0.32
ALDH1A1 P00352 1/20 0.32
GAA P10253 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28036227 0.88 SLC6A3 (0.34) SLC6A3KDM4EPKM
SCHEMBL28036658 0.88 KDM4E (0.32) KDM4EPKM
SCHEMBL27743650 0.87 SLC6A3 (0.43) SLC6A3KDM4EPKMHTT
SCHEMBL27764214 0.86 SLC6A3 (0.33) SLC6A3LMNA
SCHEMBL27741460 0.86 LY96 (0.34) SLC6A3KDM4EPKM
SCHEMBL27743460 0.86 SLC6A3 (0.33) SLC6A3FFAR1
SCHEMBL27764217 0.83 SLC6A3 (0.34) SLC6A3FFAR1CYP19A1
SCHEMBL28036656 0.79 SLC6A3 (0.36) SLC6A3CYP19A1MAPT
SCHEMBL27743428 0.78 NAMPT (0.37) SLC6A3SLC6A4KDM4ELMNA
SCHEMBL28036657 0.76 SLC6A3 (0.35) SLC6A3CYP19A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105017242-A Novel biphenyl heterocyclic derivative, preparation method and use thereof as drug UNIV CHINA PHARMA 2015-11-04 CN disclosed