SCHEMBL28038019

SCHEMBL28038019

CCn1cnc2cnc(NCc3ccccc3)nc21

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TMIGD3 P0DMS9 4/20 0.50
ADORA2A P29274 4/20 0.50
ADORA1 P30542 4/20 0.50
ALDH1A1 P00352 4/20 0.49
CYP1A2 P05177 4/20 0.49
CYP3A4 P08684 4/20 0.49
CYP2C19 P33261 4/20 0.49
HSD17B10 Q99714 4/20 0.49
CYP2D6 P10635 3/20 0.49
CYP2C9 P11712 3/20 0.49
HPGD P15428 3/20 0.49
TSHR P16473 3/20 0.49
CASP1 P29466 3/20 0.49
CASP7 P55210 3/20 0.49
ADORA2B P29275 2/20 0.49
MAPK1 P28482 2/20 0.49
HIF1A Q16665 1/20 0.49
KDM4E B2RXH2 1/20 0.46
NPC1 O15118 1/20 0.46
MAPT P10636 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8674551 0.83 CDK1 (0.59) TMIGD3ADORA2AADORA1ALDH1A1CYP1A2
SCHEMBL5335413 0.80 TDP1 (0.67) CYP1A2CYP3A4CYP2D6CYP2C9TSHR
SCHEMBL8826403 0.78 CYP1A2 (0.41) TMIGD3ADORA2AADORA1ALDH1A1CYP1A2
SCHEMBL18520823 0.78 CDK1 (0.53) TMIGD3ADORA2AADORA1ALDH1A1CYP1A2
SCHEMBL6670712 0.76 TMIGD3 (0.53) TMIGD3ADORA2AADORA1ALDH1A1CYP1A2
SCHEMBL5162419 0.76 ADORA2A (0.82) TMIGD3ADORA2AADORA1ADORA2BKDM4E
SCHEMBL22571186 0.73 TMIGD3 (0.81) TMIGD3ADORA2AADORA1HPGDADORA2B
SCHEMBL20350685 0.73 CDK1 (0.73) TMIGD3ADORA2AADORA1CYP2C19CYP2D6
SCHEMBL17450128 0.73 CDK1 (0.60) TMIGD3ADORA2AADORA1ADORA2BKDM4E
SCHEMBL28233423 0.72 ALDH1A1 (0.53) ALDH1A1CYP1A2CYP3A4CYP2C19HSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-104936959-B 2,6, 9-trisubstituted purine derivative and preparation method and application thereof 中国人民解放军军事医学科学院放射与辐射医学研究所 2018-09-18 CN disclosed
CN-104936959-A 2,6, 9-trisubstituted purine derivative and preparation method and application thereof INST RADIATION MED AMMS PLA 2015-09-23 CN disclosed