SCHEMBL28038780

SCHEMBL28038780

O=C(O)[C@@H]1CNc2ccccc2C1

nearest known ligand 0.60

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GAA P10253 1/20 0.54
MAPT P10636 1/20 0.54
MTNR1A P48039 1/20 0.50
MTNR1B P49286 1/20 0.50
EPHX2 P34913 1/20 0.48
MEN1 O00255 1/20 0.40
KMT2A Q03164 1/20 0.40
ALDH1A1 P00352 1/20 0.39
BRD4 O60885 1/20 0.38
CREBBP Q92793 1/20 0.38
IDH1 O75874 2/20 0.37
FAAH O00519 1/20 0.37
MCL1 Q07820 1/20 0.37
SMN1; SMN2 Q16637 1/20 0.37
ALOX15 P16050 1/20 0.36
HSD17B10 Q99714 1/20 0.36
AKR1C3 P42330 1/20 0.36
AKR1C1 Q04828 1/20 0.36
GABRP O00591 1/20 0.36
GABRD O14764 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30288898 1.00 GAA (0.54) GAAMAPTMTNR1AMTNR1BEPHX2
SCHEMBL924219 1.00 GAA (0.54) GAAMAPTMTNR1AMTNR1BEPHX2
SCHEMBL8562595 1.00 GAA (0.54) GAAMAPTMTNR1AMTNR1BEPHX2
SCHEMBL29463686 1.00 GAA (0.54) GAAMAPTMTNR1AMTNR1BEPHX2
SCHEMBL28114454 0.98 GAA (0.53) GAAMAPTMTNR1AMTNR1BEPHX2
Tert-Butylamine SCHEMBL28768909 0.91 EPHX2 (0.51) GAAMAPTMTNR1AMTNR1BEPHX2
SCHEMBL8901298 0.85 GAA (0.47) GAAMAPTMTNR1AMTNR1BEPHX2
SCHEMBL6419360 0.84 MTNR1A (0.49) GAAMAPTMTNR1AMTNR1BEPHX2
SCHEMBL31181154 0.84 MTNR1A (0.49) GAAMAPTMTNR1AMTNR1BEPHX2
SCHEMBL8562039 0.84 MTNR1A (0.56) GAAMAPTMTNR1AMTNR1BEPHX2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-111254181-B Method for preparing (S) -1,2,3, 4-tetrahydroisoquinoline-3-formic acid by chemical enzyme method 苏州同力生物医药有限公司 2023-06-06 CN disclosed
CN-111254170-B Method for preparing (S) -1,2,3, 4-tetrahydroisoquinoline-3-formic acid by multienzyme coupling 浙江大学 2023-04-28 CN disclosed
CN-111254180-B Method for preparing (S) -1,2,3, 4-tetrahydroisoquinoline-3-formic acid by enzymatic resolution 浙江大学 2023-04-28 CN disclosed
CN-111254180-A Method for preparing (S) -1,2,3, 4-tetrahydroisoquinoline-3-formic acid by enzymatic resolution 浙江大学 2020-06-09 CN disclosed
CN-111254170-A Method for preparing (S) -1,2,3, 4-tetrahydroisoquinoline-3-formic acid by multi-enzyme coupling 浙江大学 2020-06-09 CN disclosed
CN-111254181-A Method for preparing (S) -1,2,3, 4-tetrahydroisoquinoline-3-formic acid by chemoenzymatic method 苏州同力生物医药有限公司 2020-06-09 CN disclosed
CN-104945345-A Chiral morpholine compounds and preparation method thereof as well as chiral amino acid compounds and preparation method and application thereof SHENZHEN NEPTUNUS INTERLONG BIO TECH CO LTD 2015-09-30 CN disclosed