SCHEMBL28040110

SCHEMBL28040110

COc1ccc(Cc2cncc(N)n2)cc1

nearest known ligand 0.51

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.51
CYP2D6 P10635 1/20 0.51
ATM Q13315 1/20 0.51
POLB P06746 1/20 0.48
LTA4H P09960 2/20 0.46
LMNA P02545 1/20 0.45
HPGD P15428 1/20 0.45
NPSR1 Q6W5P4 1/20 0.44
CYP11B1 P15538 4/20 0.44
CYP11B2 P19099 4/20 0.44
MPO P05164 1/20 0.44
TLR8 Q9NR97 1/20 0.43
TLR7 Q9NYK1 1/20 0.43
SLC6A4 P31645 1/20 0.42
IDO1 P14902 1/20 0.41
AGXT P21549 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7798261 0.79 ALDH1A1 (0.53) ALDH1A1CYP2D6ATMPOLBLTA4H
SCHEMBL9391584 0.78 GRM4 (0.43) ALDH1A1LTA4HTLR8TLR7
SCHEMBL481902 0.77 ALDH1A1 (0.59) ALDH1A1CYP2D6ATMPOLBLTA4H
SCHEMBL30366498 0.75 ALDH1A1 (0.65) ALDH1A1CYP2D6ATMPOLBLTA4H
SCHEMBL28283248 0.74 CYP11B1 (0.39) ALDH1A1CYP2D6ATMPOLBLTA4H
SCHEMBL28172483 0.73 RAB9A (0.50) ALDH1A1CYP2D6ATMPOLBLTA4H
SCHEMBL29393410 0.73 ALDH1A1 (0.50) ALDH1A1CYP2D6ATMPOLBLTA4H
SCHEMBL28039277 0.73 ALDH1A1 (0.50) ALDH1A1CYP2D6ATMPOLBLTA4H
SCHEMBL28047019 0.72 ALDH1A1 (0.46) ALDH1A1CYP2D6ATMLTA4HLMNA
SCHEMBL4439445 0.71 ALDH1A1 (0.51) ALDH1A1CYP2D6ATMPOLBLTA4H

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105008367-A Pyrrolotriazines as potassium ion channel inhibitors BRISTOL MYERS SQUIBB CO 2015-10-28 CN disclosed