SCHEMBL28040158

SCHEMBL28040158

O=S(=O)(c1ccccc1)c1ncnc2[nH]ccc12

nearest known ligand 0.53

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
EGFR P00533 1/20 0.53
AURKB Q96GD4 1/20 0.53
JAK2 O60674 4/20 0.51
TTBK1 Q5TCY1 2/20 0.49
TTBK2 Q6IQ55 2/20 0.49
IKBKB O14920 2/20 0.48
CHUK O15111 2/20 0.48
TRPA1 O75762 1/20 0.48
JAK1 P23458 3/20 0.46
TYK2 P29597 2/20 0.46
JAK3 P52333 2/20 0.46
MET P08581 1/20 0.46
TNNI3K Q59H18 4/20 0.45
BRAF P15056 1/20 0.45
CDC7 O00311 1/20 0.44
DBF4 Q9UBU7 1/20 0.44
CSF1R P07333 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21218364 0.76 EGFR (0.76) EGFRAURKBJAK2TTBK1TTBK2
SCHEMBL5137242 0.75 MET (0.64) EGFRAURKBJAK2IKBKBCHUK
SCHEMBL16897037 0.72 MET (0.49) EGFRAURKBJAK2IKBKBCHUK
SCHEMBL17113647 0.72 MET (0.49) EGFRAURKBJAK1MET
SCHEMBL15542706 0.72 FFAR2 (0.44) EGFRAURKBJAK2TTBK1TTBK2
SCHEMBL16897006 0.69 MET (0.46) EGFRAURKBJAK2IKBKBCHUK
SCHEMBL5998976 0.69 HIF1A (0.48) EGFRTNNI3KBRAFCDC7DBF4
SCHEMBL19641706 0.69 FFAR2 (0.41) EGFRAURKBIKBKBCHUKMET
SCHEMBL12613146 0.68 IKBKB (0.36) EGFRAURKBJAK2IKBKBCHUK
SCHEMBL4006751 0.68 JAK2 (1.00) AURKBJAK2TTBK1TTBK2IKBKB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105189512-A Pyrrolopyrimindine CDK9 kinase inhibitors ABBVIE INC 2015-12-23 CN disclosed