SCHEMBL28040760

SCHEMBL28040760

O=C(O)C1(c2ccncc2[N+](=O)[O-])CC1

nearest known ligand 0.43

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.43
KMT2A Q03164 3/20 0.40
MEN1 O00255 2/20 0.40
HTT P42858 4/20 0.38
RAB9A P51151 1/20 0.38
MAPT P10636 4/20 0.38
HIPK2 Q9H2X6 1/20 0.36
GAA P10253 2/20 0.36
CYP1A2 P05177 1/20 0.36
CYP2C9 P11712 1/20 0.36
LMNA P02545 1/20 0.36
POLB P06746 1/20 0.36
NCOA1 Q15788 1/20 0.35
SMN1; SMN2 Q16637 1/20 0.35
NCOA3 Q9Y6Q9 1/20 0.35
PDE7A Q13946 1/20 0.35
L3MBTL1 Q9Y468 1/20 0.35
KDM4E B2RXH2 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16485964 0.84 HTT (0.43) ALDH1A1KMT2AMEN1HTTRAB9A
SCHEMBL5369495 0.79 AKR1C1 (0.46) ALDH1A1KMT2AMEN1MAPTGAA
SCHEMBL30937544 0.79 AKR1C1 (0.46) ALDH1A1KMT2AMEN1MAPTGAA
SCHEMBL14938432 0.76 MEN1 (0.42) ALDH1A1KMT2AMEN1MAPTGAA
SCHEMBL31445078 0.76 GAA (0.37) ALDH1A1KMT2AMEN1MAPTGAA
SCHEMBL28040741 0.76 KDM4E (0.49) ALDH1A1KMT2AMEN1MAPTGAA
SCHEMBL17241125 0.75 CYP1A2 (0.49) ALDH1A1KMT2AMEN1MAPTGAA
SCHEMBL5368690 0.74 AKR1C1 (0.49) ALDH1A1KMT2AMEN1MAPTGAA
SCHEMBL31447055 0.72 HDAC4 (0.39) GAAPOLB
SCHEMBL16515363 0.72 ALDH1A1 (0.39) ALDH1A1KMT2AMEN1HTTRAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105431419-A Novel aza-oxo-indoles for the treatment and prophylaxis of respiratory syncytial virus infection HOFFMANN-LA ROCHE AG 2016-03-23 CN disclosed
CN-105408330-A Novel aza-oxo-indoles for the treatment and prophylaxis of respiratory syncytial virus infection HOFFMANN LA ROCHE 2016-03-16 CN disclosed