SCHEMBL28040902

SCHEMBL28040902

O=COCCc1ncc(-c2ccccc2)s1

nearest known ligand 0.51

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
ERCC5 P28715 1/20 0.51
FEN1 P39748 1/20 0.51
LOXL2 Q9Y4K0 3/20 0.48
LOXL3 P58215 1/20 0.40
QPCT Q16769 1/20 0.39
GSTO1 P78417 1/20 0.39
KDR P35968 8/20 0.39
CCNE1 P24864 1/20 0.38
CDK2 P24941 1/20 0.38
CDK5 Q00535 1/20 0.38
ACP1 P24666 1/20 0.36
HTR7 P34969 1/20 0.36
SCD O00767 1/20 0.35
HDAC4 P56524 1/20 0.34
HDAC6 Q9UBN7 1/20 0.34
MKNK1 Q9BUB5 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28306284 0.82 MMP2 (0.38) ERCC5FEN1HDAC6
SCHEMBL13680965 0.80 ERCC5 (0.55) ERCC5FEN1LOXL2LOXL3QPCT
SCHEMBL31595961 0.76 ERCC5 (0.58) ERCC5FEN1LOXL2LOXL3QPCT
SCHEMBL28003535 0.75 HDAC6 (0.46) QPCTHDAC6
SCHEMBL2227416 0.74 LOXL2 (0.64) ERCC5FEN1LOXL2LOXL3QPCT
SCHEMBL28815683 0.74 LOXL2 (0.55) ERCC5FEN1LOXL2LOXL3QPCT
SCHEMBL28602757 0.73
SCHEMBL4873585 0.72 LOXL2 (0.53) ERCC5FEN1LOXL2LOXL3QPCT
SCHEMBL5677058 0.72 LOXL2 (0.49) ERCC5FEN1LOXL2LOXL3QPCT
SCHEMBL25523340 0.71 LOXL2 (0.51) ERCC5FEN1LOXL2LOXL3QPCT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105228982-A 3-acetylamino-1- (phenyl-heteroaryl-aminocarbonyl or phenyl-heteroaryl-carbonylamino) benzene derivatives for the treatment of hyperproliferative disorders Bayer Pharma AG 2016-01-06 CN disclosed