SCHEMBL28041598

SCHEMBL28041598

Nc1nc2ccccc2c(-c2ccccc2)c1-c1ccccc1

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 6/20 0.56
MAPT P10636 5/20 0.56
TDP1 Q9NUW8 2/20 0.56
MAPK1 P28482 1/20 0.56
L3MBTL1 Q9Y468 1/20 0.56
ESR1 P03372 4/20 0.52
ESR2 Q92731 4/20 0.52
ALDH1A1 P00352 5/20 0.50
HSD17B10 Q99714 5/20 0.50
HPGD P15428 4/20 0.50
GAA P10253 3/20 0.50
ACHE P22303 2/20 0.50
GLA P06280 2/20 0.50
CASP1 P29466 2/20 0.50
CASP7 P55210 2/20 0.50
SMN1; SMN2 Q16637 2/20 0.50
CHRM2 P08172 1/20 0.50
ADRA2A P08913 1/20 0.50
ADORA3 P0DMS8 1/20 0.50
CHRM1 P11229 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5080981 0.86 KDM4E (0.59) KDM4EMAPTTDP1MAPK1L3MBTL1
SCHEMBL27590144 0.83 NPC1 (0.50) KDM4EMAPTTDP1MAPK1L3MBTL1
SCHEMBL4263725 0.82 MAPT (0.47) KDM4EMAPTTDP1MAPK1L3MBTL1
SCHEMBL11576048 0.82 KDM4E (0.51) KDM4EMAPTTDP1MAPK1L3MBTL1
SCHEMBL28041606 0.81 KDM4E (0.47) KDM4EMAPTTDP1MAPK1L3MBTL1
SCHEMBL29514776 0.80 ESR1 (0.73) KDM4EMAPTTDP1ESR1ESR2
SCHEMBL194068 0.80 ESR1 (0.73) KDM4EMAPTTDP1ESR1ESR2
SCHEMBL6220647 0.80 DPP4 (0.59) KDM4EMAPTTDP1MAPK1L3MBTL1
SCHEMBL4436700 0.78 ADORA2A (0.60) KDM4EMAPTALDH1A1HSD17B10HPGD
SCHEMBL28823862 0.78 FABP4 (0.54) KDM4EMAPTMAPK1ESR1ESR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-104086485-B Prepare the method for poly-substituted quinoline type aromatic ring pyridine derivate TSINGHUA UNIVERSITY (CN) 2016-03-30 CN disclosed