SCHEMBL28041982

SCHEMBL28041982

O=C1CCN(C(F)c2ccccc2)CC1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP2D6 P10635 6/20 0.39
KCNH2 Q12809 5/20 0.39
CYP1A2 P05177 4/20 0.39
CYP3A4 P08684 4/20 0.39
CYP2C9 P11712 4/20 0.39
KCNA5 P22460 4/20 0.39
CYP2C19 P33261 4/20 0.39
KCNE1 P15382 1/20 0.38
HSD11B1 P28845 2/20 0.37
LMNA P02545 1/20 0.37
TACR1 P25103 3/20 0.36
KMT2A Q03164 2/20 0.36
CHRM2 P08172 1/20 0.36
CHRM4 P08173 1/20 0.36
CHRM5 P08912 1/20 0.36
ADRA2A P08913 1/20 0.36
ADORA3 P0DMS8 1/20 0.36
CHRM1 P11229 1/20 0.36
CHRM3 P20309 1/20 0.36
DRD1 P21728 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5391913 0.80 KMT2A (0.57) CYP2D6KCNH2CYP2C19KMT2ACHRM2
SCHEMBL3208256 0.78 CYP1A2 (0.63) CYP2D6KCNH2CYP1A2CYP3A4CYP2C9
SCHEMBL1586528 0.77 CYP2D6 (0.70) CYP2D6HSD11B1CHRM2CHRM1OPRM1
SCHEMBL19631646 0.77 TACR1 (0.40) CYP2D6KCNH2CYP1A2CYP3A4CYP2C9
SCHEMBL28041843 0.77 CYP2D6 (0.39) CYP2D6KCNH2CYP1A2CYP3A4CYP2C9
SCHEMBL19613500 0.77 CYP2D6 (0.70) CYP2D6HSD11B1CHRM2CHRM1OPRM1
SCHEMBL4601165 0.77 CYP2D6 (0.70) CYP2D6HSD11B1CHRM2CHRM1OPRM1
SCHEMBL8099850 0.77 CYP2D6 (0.70) CYP2D6HSD11B1CHRM2CHRM1OPRM1
SCHEMBL4696100 0.77 CYP2D6 (0.39) CYP2D6KCNH2CYP1A2CYP3A4CYP2C9
SCHEMBL27330921 0.77 LMNA (0.41) CYP2D6KCNH2CYP1A2CYP3A4CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-103288824-B Tetrahydropyridine Pyridione derivatives, its preparation method and application SHANGHAI NORMAL UNIVERSITY (CN) 2015-12-09 CN disclosed