SCHEMBL28042358

SCHEMBL28042358

CCC(=O)N1CCC(c2cnc(N)c(OC(C)=O)n2)CC1

nearest known ligand 0.38

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
MAP3K12 Q12852 1/20 0.38
TRPC6 Q9Y210 1/20 0.37
PIK3CD O00329 10/20 0.37
MAPK1 P28482 3/20 0.37
PIK3R1 P27986 1/20 0.36
RIPK1 Q13546 1/20 0.36
MET P08581 1/20 0.35
KDR P35968 2/20 0.35
PIK3CA P42336 2/20 0.35
PIK3CB P42338 2/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27875132 0.84 ATR (0.40) MAP3K12MAPK1
SCHEMBL28076399 0.81 EPHX2 (0.39) MAP3K12TRPC6MAPK1RIPK1MET
SCHEMBL617266 0.81 ATR (0.42) MAP3K12TRPC6PIK3CDMAPK1
SCHEMBL28042583 0.78 HRH4 (0.38) MAPK1MET
SCHEMBL28042359 0.78 MAPKAPK2 (0.39) MAP3K12TRPC6PIK3CDMAPK1RIPK1
SCHEMBL615145 0.78 ATR (0.47) TRPC6PIK3CDMAPK1
SCHEMBL28776119 0.69 MAPT (0.44) MAPK1
SCHEMBL16678995 0.69 MAPK1 (0.44) MAP3K12PIK3CDMAPK1
SCHEMBL27926722 0.69 TRPC6 (0.51) TRPC6RIPK1
SCHEMBL28042291 0.69 EPHX2 (0.38) TRPC6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-102264721-B Compounds useful as inhibitors of ATR kinase VERTEX PHARMACEUTICALS INC. (US) 2015-12-09 CN disclosed