SCHEMBL28042291

SCHEMBL28042291

CCC(=O)N1CCC(c2cnc(N)cn2)CC1.NNC=O

nearest known ligand 0.38

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
EPHX2 P34913 9/20 0.38
TRPC6 Q9Y210 4/20 0.38
CHEK1 O14757 1/20 0.35
PDCD1 Q15116 1/20 0.35
CD274 Q9NZQ7 1/20 0.35
TLR9 Q9NR96 2/20 0.35
TLR8 Q9NR97 2/20 0.35
TLR7 Q9NYK1 2/20 0.35
CHRM4 P08173 1/20 0.35
CHRM1 P11229 1/20 0.35
JAK1 P23458 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21275520 0.76 TRPC6 (0.37) TRPC6
SCHEMBL615145 0.74 ATR (0.47) EPHX2TRPC6
SCHEMBL27926722 0.73 TRPC6 (0.51) EPHX2TRPC6TLR9TLR8TLR7
SCHEMBL28076399 0.72 EPHX2 (0.39) EPHX2TRPC6
SCHEMBL617266 0.72 ATR (0.42) EPHX2TRPC6
SCHEMBL15175760 0.71 GPR119 (0.54) JAK1
SCHEMBL28042359 0.70 MAPKAPK2 (0.39) EPHX2TRPC6
SCHEMBL28042358 0.69 MAP3K12 (0.38) TRPC6
SCHEMBL28776119 0.68 MAPT (0.44) EPHX2
SCHEMBL26157258 0.67 PIK3CD (0.46) EPHX2TLR9TLR8TLR7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-102264721-B Compounds useful as inhibitors of ATR kinase VERTEX PHARMACEUTICALS INC. (US) 2015-12-09 CN disclosed