SCHEMBL28043557

SCHEMBL28043557

Nc1cccc(Cc2cccnc2)n1

nearest known ligand 0.50

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
CHRNA7 P36544 1/20 0.46
MPO P05164 1/20 0.46
CYP1A2 P05177 2/20 0.44
CYP2D6 P10635 2/20 0.44
HRH4 Q9H3N8 1/20 0.44
HRH3 Q9Y5N1 1/20 0.44
CYP2A6 P11509 1/20 0.43
ADORA2A P29274 1/20 0.42
ALDH1A1 P00352 1/20 0.41
PKM P14618 1/20 0.41
MMP2 P08253 1/20 0.41
HRH1 P35367 2/20 0.41
LTA4H P09960 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28043533 0.80 CYP17A1 (0.47) ADORA2A
SCHEMBL29758354 0.80 BACE1 (0.50) ADORA2AALDH1A1
SCHEMBL1402167 0.80 BACE1 (0.50) ADORA2AALDH1A1
SCHEMBL7969373 0.79 CYP1A2 (0.44) CHRNA7CYP1A2CYP2D6HRH4HRH3
SCHEMBL19591018 0.79 CYP2A6 (0.49) CHRNA7CYP1A2CYP2D6HRH4HRH3
SCHEMBL28108406 0.76 PDE10A (0.47) CHRNA7MPOCYP1A2CYP2D6HRH4
SCHEMBL29520054 0.75 CHRNA7 (0.44) CHRNA7MPOCYP1A2CYP2D6HRH4
SCHEMBL727185 0.74 CYP1A2 (0.62) CHRNA7CYP1A2CYP2D6HRH4HRH3
SCHEMBL4938657 0.74 BACE1 (0.62) CYP1A2CYP2D6CYP2A6ADORA2AALDH1A1
SCHEMBL17674597 0.73 GAA (0.41) CHRNA7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105324380-A Pyrrolo[2,3-b]pyridine cdk9 kinase inhibitors ABBVIE INC 2016-02-10 CN disclosed
CN-105246890-A Pyrrolo[2, 3-b]pyridine cdk9 kinase inhibitors ABBVIE INC 2016-01-13 CN disclosed