SCHEMBL28043769

SCHEMBL28043769

CCCCc1c(N)nc(N)nc1-c1cccc(Cl)c1

nearest known ligand 0.55

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
DHFR P00374 4/20 0.54
ADORA2A P29274 4/20 0.51
ADORA1 P30542 4/20 0.51
ADORA2B P29275 2/20 0.51
DPP4 P27487 1/20 0.50
MAP4K4 O95819 2/20 0.47
TLR8 Q9NR97 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28043971 0.83 HEXA (0.55) DHFRADORA2AADORA1DPP4TLR8
SCHEMBL28043777 0.81 ADORA2A (0.51) DHFRADORA2AADORA1DPP4TLR8
Hydrochloric Acid SCHEMBL20421687 0.80 TLR8 (0.48) DHFRTLR8
SCHEMBL22139488 0.78 DHFR (0.54) DHFRADORA2AADORA1ADORA2B
SCHEMBL28043715 0.77 CYP2D6 (0.52) DHFR
SCHEMBL28043944 0.77 HEXA (0.50) DHFRADORA2AADORA1TLR8
SCHEMBL29913459 0.76 DHFR (0.74) DHFR
SCHEMBL12495851 0.75 TLR8 (0.60) DHFRADORA2AADORA1ADORA2BTLR8
SCHEMBL12495846 0.74 TLR8 (0.54) DHFRADORA2AADORA1TLR8
SCHEMBL4418415 0.74 ADORA2A (0.59) DHFRADORA2AADORA1ADORA2BDPP4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105143206-A Pyrimidine-2,4-diamine derivatives for treatment of cancer THOMAS HELLEDAYS STIFTELSE F R MEDICINSK FORSKNING 2015-12-09 CN disclosed