SCHEMBL28043944

SCHEMBL28043944

CCCCc1c(N)nc(N)nc1-c1cc(C)cc(C)c1

nearest known ligand 0.50

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
HEXA P06865 3/20 0.50
HEXB P07686 3/20 0.50
NOS2 P35228 2/20 0.46
ADORA2A P29274 1/20 0.42
ADORA1 P30542 1/20 0.42
ALDH1A1 P00352 1/20 0.40
MAPT P10636 1/20 0.40
KMT2A Q03164 1/20 0.40
CYP2D6 P10635 1/20 0.39
TLR8 Q9NR97 5/20 0.39
TLR7 Q9NYK1 1/20 0.39
DHFR P00374 2/20 0.38
NOS3 P29474 1/20 0.38
NOS1 P29475 1/20 0.38
HRH2 P25021 1/20 0.38
HRH3 Q9Y5N1 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29262764 0.78 CYP2D6 (0.52) NOS2ALDH1A1MAPTKMT2ACYP2D6
SCHEMBL28043971 0.78 HEXA (0.55) HEXAHEXBADORA2AADORA1ALDH1A1
SCHEMBL16703398 0.78 DHFR (0.43) CYP2D6TLR8TLR7DHFR
SCHEMBL28043769 0.77 DHFR (0.54) ADORA2AADORA1TLR8DHFR
SCHEMBL28043777 0.74 ADORA2A (0.51) HEXAHEXBADORA2AADORA1CYP2D6
SCHEMBL6345470 0.73 KMT2A (0.47) HEXAHEXBNOS2ALDH1A1MAPT
SCHEMBL20242690 0.73 TLR8 (0.59) TLR8TLR7DHFR
SCHEMBL30035562 0.73 TLR8 (0.59) TLR8TLR7DHFR
Hydrochloric Acid SCHEMBL20421687 0.73 TLR8 (0.48) CYP2D6TLR8DHFR
SCHEMBL4463336 0.73 HEXA (0.47) HEXAHEXBADORA2AADORA1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105143206-A Pyrimidine-2,4-diamine derivatives for treatment of cancer THOMAS HELLEDAYS STIFTELSE F R MEDICINSK FORSKNING 2015-12-09 CN disclosed