SCHEMBL28043877

SCHEMBL28043877

NCc1cccc(-c2cc(Cl)nc(N)n2)c1Cl

nearest known ligand 0.59

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HSP90AA1 P07900 9/20 0.59
HSP90AB1 P08238 9/20 0.59
KDM4E B2RXH2 1/20 0.50
NUDT1 P36639 2/20 0.47
PDCD1LG2 Q9BQ51 1/20 0.47
CD274 Q9NZQ7 1/20 0.47
ADCY10 Q96PN6 6/20 0.44
CDC7 O00311 1/20 0.44
DAPK3 O43293 1/20 0.44
PRKD3 O94806 1/20 0.44
MAP4K4 O95819 1/20 0.44
PAK4 O96013 1/20 0.44
PIM1 P11309 1/20 0.44
PRKACA P17612 1/20 0.44
GRK5 P34947 1/20 0.44
MAP2K2 P36507 1/20 0.44
MAPK8 P45983 1/20 0.44
CSNK1A1 P48729 1/20 0.44
CDK8 P49336 1/20 0.44
CLK2 P49760 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3952703 0.84 HSP90AA1 (0.52) HSP90AA1HSP90AB1KDM4ENUDT1ADCY10
SCHEMBL4281168 0.82 HSP90AA1 (0.75) HSP90AA1HSP90AB1KDM4ENUDT1ADCY10
SCHEMBL28043746 0.81 NUDT1 (0.73) HSP90AA1HSP90AB1NUDT1PDCD1LG2CD274
SCHEMBL28043914 0.80 HSP90AA1 (0.67) HSP90AA1HSP90AB1KDM4ENUDT1ADCY10
SCHEMBL3945480 0.79 HSP90AA1 (0.61) HSP90AA1HSP90AB1KDM4ENUDT1ADCY10
SCHEMBL28043754 0.78 HSP90AB1 (0.62) HSP90AA1HSP90AB1KDM4EADCY10CDC7
SCHEMBL28043721 0.77 NUDT1 (0.76) NUDT1PDCD1LG2CD274ROCK1
SCHEMBL28265686 0.76 CD274 (0.44) PDCD1LG2CD274CDC7DAPK3MAP4K4
SCHEMBL3952031 0.76 HSP90AA1 (0.78) HSP90AA1HSP90AB1KDM4ENUDT1ADCY10
SCHEMBL15757653 0.75 HSP90AA1 (0.67) HSP90AA1HSP90AB1KDM4ENUDT1CDC7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105143206-A Pyrimidine-2,4-diamine derivatives for treatment of cancer THOMAS HELLEDAYS STIFTELSE F R MEDICINSK FORSKNING 2015-12-09 CN disclosed