SCHEMBL28265686

SCHEMBL28265686

NCc1cccc(-c2cc(Cl)ncn2)c1Cl

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CD274 Q9NZQ7 6/20 0.44
PDCD1LG2 Q9BQ51 2/20 0.44
PNMT P11086 2/20 0.43
CLK4 Q9HAZ1 4/20 0.41
CDC7 O00311 1/20 0.41
DAPK3 O43293 1/20 0.41
MAP4K4 O95819 1/20 0.41
PIM1 P11309 1/20 0.41
PRKACA P17612 1/20 0.41
FLT3 P36888 1/20 0.41
CDK8 P49336 1/20 0.41
CLK2 P49760 1/20 0.41
GSK3B P49841 1/20 0.41
CDK7 P50613 1/20 0.41
CDK9 P50750 1/20 0.41
PRKX P51817 1/20 0.41
CDK5 Q00535 1/20 0.41
DYRK1A Q13627 1/20 0.41
PKN2 Q16513 1/20 0.41
MINK1 Q8N4C8 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28265660 0.80 IDO1 (0.46) CLK4CDC7DAPK3MAP4K4PIM1
SCHEMBL28267446 0.79 CLK4 (0.40) PNMTCLK4CDC7DAPK3MAP4K4
SCHEMBL28267174 0.77 CDC7 (0.38) CD274PDCD1LG2CLK4CDC7DAPK3
SCHEMBL28043877 0.76 HSP90AA1 (0.59) CD274PDCD1LG2PNMTCLK4CDC7
SCHEMBL16655898 0.76 DPP4 (0.53) PNMTCLK4CDC7DAPK3MAP4K4
SCHEMBL14050408 0.75 CLK4 (0.46) CLK4CDC7DAPK3MAP4K4PIM1
SCHEMBL4436881 0.75 CYP2D6 (0.47) CLK4CDC7DAPK3MAP4K4PIM1
SCHEMBL1415582 0.73 CLK4 (0.45) CLK4CDC7DAPK3MAP4K4PIM1
SCHEMBL4429838 0.72 CYP2D6 (0.44) CLK4CDC7DAPK3MAP4K4PIM1
SCHEMBL28151150 0.70 IDO1 (0.49) CLK4CDC7DAPK3MAP4K4PIM1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105143206-B Pyrimidine -2,4- diamine derivative for treating cancer 托马斯·黑勒戴药物研究基金会 2019-01-15 CN disclosed