SCHEMBL28043933

SCHEMBL28043933

Cc1cc(C)cc(-c2cc(NCCc3ccc(CN)cc3)nc(N)n2)c1

nearest known ligand 0.50

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
HRH4 Q9H3N8 10/20 0.50
TLR8 Q9NR97 1/20 0.47
ALDH1A1 P00352 1/20 0.47
SMN1; SMN2 Q16637 1/20 0.47
PTGDR Q13258 7/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28151182 0.92 HRH4 (0.52) HRH4TLR8ALDH1A1SMN1; SMN2PTGDR
SCHEMBL28043774 0.89 HRH4 (0.49) HRH4TLR8ALDH1A1SMN1; SMN2PTGDR
SCHEMBL28043806 0.89 ALDH1A1 (0.52) HRH4TLR8ALDH1A1SMN1; SMN2PTGDR
SCHEMBL28043771 0.89 HRH4 (0.62) HRH4TLR8ALDH1A1SMN1; SMN2PTGDR
SCHEMBL28043714 0.88 HRH4 (0.50) HRH4TLR8ALDH1A1SMN1; SMN2PTGDR
SCHEMBL28267214 0.87 PTGDR (0.57) PTGDR
SCHEMBL28152055 0.86 PTGDR (0.48) HRH4TLR8ALDH1A1SMN1; SMN2PTGDR
SCHEMBL28151132 0.85 CA1 (0.56) HRH4ALDH1A1SMN1; SMN2PTGDR
SCHEMBL28152277 0.85 HRH4 (0.48) HRH4TLR8ALDH1A1SMN1; SMN2PTGDR
SCHEMBL28151149 0.84 HRH4 (0.64) HRH4TLR8

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105143206-B Pyrimidine -2,4- diamine derivative for treating cancer 托马斯·黑勒戴药物研究基金会 2019-01-15 CN claimed
CN-105143206-B Pyrimidine -2,4- diamine derivative for treating cancer 托马斯·黑勒戴药物研究基金会 2019-01-15 CN disclosed
CN-106794181-A MTH1 inhibitors for the treatment of inflammatory and autoimmune conditions 托马斯·黑勒戴药物研究基金会 2017-05-31 CN disclosed
CN-105143206-A Pyrimidine-2,4-diamine derivatives for treatment of cancer THOMAS HELLEDAYS STIFTELSE F R MEDICINSK FORSKNING 2015-12-09 CN disclosed