SCHEMBL28043993

SCHEMBL28043993

NCc1cccc(-c2cc(NCCc3ccc(Cl)cc3)nc(N)n2)c1Cl

nearest known ligand 0.50

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 1/20 0.48
SMN1; SMN2 Q16637 1/20 0.48
NUDT1 P36639 2/20 0.46
HRH4 Q9H3N8 3/20 0.43
AGPAT2 O15120 7/20 0.41
ACKR3 P25106 1/20 0.40
HTR2B P41595 1/20 0.40
PTGDR Q13258 2/20 0.40
CDK9 P50750 1/20 0.39
ADORA2A P29274 1/20 0.39
TLR8 Q9NR97 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28043805 0.92 ALDH1A1 (0.49) ALDH1A1SMN1; SMN2NUDT1HRH4AGPAT2
SCHEMBL15757477 0.89 NUDT1 (0.60) ALDH1A1SMN1; SMN2NUDT1HRH4AGPAT2
SCHEMBL15756895 0.87 NUDT1 (0.49) ALDH1A1SMN1; SMN2NUDT1HRH4AGPAT2
SCHEMBL28043953 0.86 ALDH1A1 (0.50) ALDH1A1SMN1; SMN2HRH4AGPAT2ACKR3
SCHEMBL17315288 0.84 HTR2B (0.54) ALDH1A1SMN1; SMN2HRH4AGPAT2ACKR3
SCHEMBL15757697 0.83 ALDH1A1 (0.54) ALDH1A1SMN1; SMN2NUDT1HRH4AGPAT2
SCHEMBL15757676 0.82 NUDT1 (0.59) ALDH1A1SMN1; SMN2NUDT1HRH4AGPAT2
SCHEMBL17315523 0.82 NUDT1 (0.49) ALDH1A1SMN1; SMN2NUDT1HRH4AGPAT2
SCHEMBL15757319 0.82 AGPAT2 (0.53) ALDH1A1SMN1; SMN2NUDT1HRH4AGPAT2
SCHEMBL17315254 0.81 ALDH1A1 (0.58) ALDH1A1SMN1; SMN2HRH4AGPAT2ACKR3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105143206-B Pyrimidine -2,4- diamine derivative for treating cancer 托马斯·黑勒戴药物研究基金会 2019-01-15 CN claimed
CN-105143206-B Pyrimidine -2,4- diamine derivative for treating cancer 托马斯·黑勒戴药物研究基金会 2019-01-15 CN disclosed
CN-105143206-A Pyrimidine-2,4-diamine derivatives for treatment of cancer THOMAS HELLEDAYS STIFTELSE F R MEDICINSK FORSKNING 2015-12-09 CN disclosed