SCHEMBL28044048

SCHEMBL28044048

COc1ccccc1-c1ccn(C(c2ccccc2)(c2ccccc2)c2ccccc2)n1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
METAP2 P50579 1/20 0.42
MAPT P10636 3/20 0.41
ALDH1A1 P00352 5/20 0.41
KDM4E B2RXH2 2/20 0.41
GAA P10253 2/20 0.41
POLB P06746 1/20 0.41
FYN P06241 2/20 0.40
JAK2 O60674 2/20 0.40
HSP90AA1 P07900 2/20 0.39
HPGD P15428 2/20 0.39
MEN1 O00255 1/20 0.39
KMT2A Q03164 1/20 0.39
NPSR1 Q6W5P4 1/20 0.39
HSD17B10 Q99714 2/20 0.39
JAK3 P52333 1/20 0.39
LMNA P02545 1/20 0.39
CYP1A2 P05177 1/20 0.39
CYP3A4 P08684 1/20 0.39
CYP2D6 P10635 1/20 0.39
TSHR P16473 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29685392 0.77 KMT2A (0.50) METAP2MAPTALDH1A1KDM4EGAA
SCHEMBL12844824 0.77 KMT2A (0.50) METAP2MAPTALDH1A1KDM4EGAA
SCHEMBL5800759 0.75 KMT2A (0.52) MAPTALDH1A1KDM4EHPGDMEN1
SCHEMBL9089445 0.75 NPC1 (0.38) MAPTALDH1A1KDM4EGAAPOLB
SCHEMBL28044043 0.74 MAOB (0.43) MAPTALDH1A1KDM4EFYNHPGD
SCHEMBL28066998 0.74 METAP2 (0.46) METAP2MAPTALDH1A1KDM4EGAA
SCHEMBL989470 0.74 GRM5 (0.40) ALDH1A1CYP3A4CYP2C19TP53
SCHEMBL11623460 0.73 ALDH1A1 (0.40) METAP2MAPTALDH1A1KDM4EFYN
SCHEMBL3852029 0.73 KDR (0.43) FYNJAK2MEN1KMT2ALMNA
SCHEMBL12777944 0.72 METAP2 (0.44) METAP2MAPTALDH1A1KDM4EGAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105050598-A Novel compounds as ERK inhibitors MERCK SHARP & DOHME 2015-11-11 CN disclosed