SCHEMBL28044154

SCHEMBL28044154

CCc1cccc(C#N)c1CCBr

nearest known ligand 0.39

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
GABRA1 P14867 4/20 0.39
GABRB2 P47870 4/20 0.39
TSHR P16473 5/20 0.34
AR P10275 1/20 0.33
CA1 P00915 1/20 0.33
CA2 P00918 1/20 0.33
NPSR1 Q6W5P4 1/20 0.32
ALDH1A1 P00352 1/20 0.32
HTR1A P08908 1/20 0.32
TAAR1 Q96RJ0 1/20 0.32
APLNR P35414 1/20 0.32
CYP2C9 P11712 1/20 0.32
S1PR1 P21453 1/20 0.32
FFAR1 O14842 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16097833 0.86 GABRA1 (0.42) GABRA1GABRB2TSHRARCA1
SCHEMBL7790350 0.83 GABRA1 (0.41) GABRA1GABRB2TSHRARCA1
SCHEMBL27367558 0.77 DYRK1A (0.40) TSHRCA1CA2
SCHEMBL25843243 0.76 AR (0.35) TSHRARALDH1A1
SCHEMBL22447106 0.75 TSHR (0.36) GABRA1GABRB2TSHRARCYP2C9
SCHEMBL16771350 0.75 TSHR (0.46) TSHRCA1CA2ALDH1A1CYP2C9
SCHEMBL8763180 0.74 GABRA1 (0.40) GABRA1GABRB2TSHRARCA1
SCHEMBL5728797 0.74 CYP19A1 (0.43) TSHRNPSR1ALDH1A1FFAR1
SCHEMBL30252315 0.74 CYP19A1 (0.43) TSHRNPSR1ALDH1A1FFAR1
SCHEMBL106062 0.73 TSHR (0.50) GABRA1GABRB2TSHRARCA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105051044-A Compounds and their use for modulating hemoglobin GLOBAL BLOOD THERAPEUTICS INC 2015-11-11 CN disclosed