SCHEMBL28044290

SCHEMBL28044290

COc1ccc2cc(C(=O)OCP(=O)(O)O)oc2c1

nearest known ligand 0.57

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 1/20 0.57
CYP2D6 P10635 2/20 0.55
ALDH1A1 P00352 4/20 0.51
HPGD P15428 4/20 0.51
KDM4E B2RXH2 4/20 0.51
GAA P10253 3/20 0.51
CA2 P00918 3/20 0.51
CA12 O43570 3/20 0.51
CA4 P22748 3/20 0.51
CA7 P43166 3/20 0.51
GLA P06280 2/20 0.51
MAOB P27338 2/20 0.51
CA3 P07451 2/20 0.51
CA6 P23280 2/20 0.51
CA9 Q16790 2/20 0.51
CA14 Q9ULX7 2/20 0.51
MAPT P10636 2/20 0.50
CASP3 P42574 1/20 0.50
SENP7 Q9BQF6 1/20 0.50
TDP1 Q9NUW8 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL177458 0.84 HPGD (0.70) CYP1A2CYP2D6ALDH1A1HPGDKDM4E
SCHEMBL28044304 0.81 CYP2D6 (0.51) CYP1A2CYP2D6ALDH1A1HPGDKDM4E
SCHEMBL4450673 0.81 KDM4E (0.67) CYP1A2CYP2D6ALDH1A1HPGDKDM4E
SCHEMBL6240000 0.78 CYP2D6 (0.70) CYP2D6ALDH1A1HPGDKDM4EGAA
SCHEMBL29233648 0.77 KDM4E (0.61) CYP1A2CYP2D6ALDH1A1HPGDKDM4E
SCHEMBL1287537 0.76 ALDH1A1 (0.66) CYP1A2CYP2D6ALDH1A1HPGDKDM4E
SCHEMBL178096 0.76 ALDH1A1 (0.66) CYP1A2CYP2D6ALDH1A1HPGDKDM4E
SCHEMBL31367874 0.76 CYP2D6 (0.59) CYP1A2CYP2D6ALDH1A1HPGDKDM4E
SCHEMBL29233580 0.76 HSD17B10 (0.64) CYP1A2CYP2D6ALDH1A1HPGDKDM4E
SCHEMBL29233642 0.75 CYP1A2 (0.84) CYP1A2CYP2D6ALDH1A1HPGDKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-103130705-B Benzo five-membered unsaturated heterocycle compound or its pharmaceutical salts and preparation method thereof, pharmaceutical composition and application thereof INSTITUTE OF MEDICINAL BIOTECHNOLOGY, CHINESE ACADEMY OF MEDICAL SCIENCES (CN) 2016-04-20 CN claimed
CN-103130705-B Benzo five-membered unsaturated heterocycle compound or its pharmaceutical salts and preparation method thereof, pharmaceutical composition and application thereof INSTITUTE OF MEDICINAL BIOTECHNOLOGY, CHINESE ACADEMY OF MEDICAL SCIENCES (CN) 2016-04-20 CN disclosed