SCHEMBL28044386

SCHEMBL28044386

COc1ccc2c(C(C)OC)c(C(=O)O)[nH]c2c1

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GPR17 Q13304 1/20 0.56
KDM4E B2RXH2 9/20 0.51
ALDH1A1 P00352 7/20 0.51
HPGD P15428 5/20 0.51
HSD17B10 Q99714 4/20 0.51
GAA P10253 4/20 0.51
MAPT P10636 3/20 0.51
ALOX15 P16050 2/20 0.51
USP2 O75604 1/20 0.51
NPSR1 Q6W5P4 1/20 0.51
KMT2A Q03164 4/20 0.49
MEN1 O00255 3/20 0.46
TDP1 Q9NUW8 2/20 0.46
GSK3A P49840 1/20 0.44
GSK3B P49841 1/20 0.44
GFER P55789 1/20 0.44
CDK5 Q00535 1/20 0.44
CDK5R1 Q15078 1/20 0.44
POLB P06746 3/20 0.44
MDM2 Q00987 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9189032 0.83 GPR17 (0.59) GPR17KDM4EALDH1A1HPGDHSD17B10
SCHEMBL1144751 0.80 GPR17 (0.64) GPR17KDM4EALDH1A1HPGDHSD17B10
SCHEMBL30779683 0.79 GPR17 (0.63) GPR17KDM4EALDH1A1HPGDHSD17B10
SCHEMBL8692433 0.78 KDM4E (0.59) GPR17KDM4EALDH1A1HPGDHSD17B10
SCHEMBL4877546 0.76 GPR17 (0.60) GPR17KDM4EALDH1A1HPGDHSD17B10
SCHEMBL29956530 0.75 GPR17 (0.59) GPR17KDM4EALDH1A1HPGDHSD17B10
SCHEMBL20535956 0.74 KDM4E (0.60) GPR17KDM4EALDH1A1HPGDHSD17B10
SCHEMBL9672508 0.74 KDM4E (0.57) GPR17KDM4EALDH1A1HPGDHSD17B10
SCHEMBL7501990 0.73 ALDH1A1 (0.65) GPR17KDM4EALDH1A1HPGDHSD17B10
SCHEMBL4878704 0.72 GPR17 (0.49) GPR17KDM4EALDH1A1HPGDHSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-103130705-B Benzo five-membered unsaturated heterocycle compound or its pharmaceutical salts and preparation method thereof, pharmaceutical composition and application thereof INSTITUTE OF MEDICINAL BIOTECHNOLOGY, CHINESE ACADEMY OF MEDICAL SCIENCES (CN) 2016-04-20 CN disclosed