SCHEMBL28046779

SCHEMBL28046779

O=C(Cc1ccccc1)NC(Cc1c[nH]c2ccccc12)C(=O)O

nearest known ligand 0.71

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
ECE1 P42892 1/20 0.71
ALOX15 P16050 1/20 0.67
LTA4H P09960 1/20 0.66
P2RY14 Q15391 1/20 0.66
ACE P12821 4/20 0.65
ITGB2 P05107 3/20 0.65
ICAM1 P05362 3/20 0.65
ITGAL P20701 3/20 0.65
POLB P06746 2/20 0.64
MEN1 O00255 1/20 0.64
HTT P42858 1/20 0.64
KMT2A Q03164 1/20 0.64
ERAP2 Q6P179 1/20 0.64
TP53 P04637 1/20 0.63

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11591677 1.00 ECE1 (0.71) ECE1ALOX15LTA4HP2RY14ACE
SCHEMBL13278205 0.92 ALOX15 (0.70) ALOX15P2RY14ACEITGB2ICAM1
SCHEMBL29987387 0.92 ALOX15 (0.70) ALOX15P2RY14ACEITGB2ICAM1
SCHEMBL3728145 0.92 ALOX15 (0.70) ALOX15P2RY14ACEITGB2ICAM1
SCHEMBL11863617 0.92 ITGB2 (0.67) ECE1ALOX15P2RY14ACEITGB2
SCHEMBL4680711 0.90 ECE1 (0.68) ECE1LTA4HP2RY14ERAP2
SCHEMBL503091 0.90 KMT2A (0.68) ECE1ALOX15LTA4HP2RY14ACE
SCHEMBL30069244 0.90 KMT2A (0.68) ECE1ALOX15LTA4HP2RY14ACE
SCHEMBL29557188 0.90 KMT2A (0.68) ECE1ALOX15LTA4HP2RY14ACE
SCHEMBL1574598 0.90 KMT2A (0.68) ECE1ALOX15LTA4HP2RY14ACE

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105198884-B Pentacyclic indole quinolizine that the G1/G0 phases block, its synthesis, antitumor activity and application 首都医科大学 2017-08-01 CN disclosed
CN-105198884-A G1/G0-phase blocked pentacyclic indol-quinolizidine and compound, antineoplastic activity and application thereof UNIV CAPITAL MEDICAL SCIENCES 2015-12-30 CN disclosed
CN-101863926-A Antitumor drug palladium coordination compound UNIV HEBEI 2010-10-20 CN disclosed