SCHEMBL28047795

SCHEMBL28047795

Nc1ncc(Cc2cccc(F)c2)nc1N

nearest known ligand 0.58

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
L3MBTL1 Q9Y468 1/20 0.43
NPC1 O15118 1/20 0.43
RAB9A P51151 1/20 0.43
MPO P05164 1/20 0.43
TAAR1 Q96RJ0 2/20 0.42
MAOB P27338 3/20 0.42
HTR2C P28335 1/20 0.41
HTR2B P41595 1/20 0.41
IDO1 P14902 2/20 0.41
AGXT P21549 2/20 0.41
APP P05067 1/20 0.41
TLR8 Q9NR97 1/20 0.40
TLR7 Q9NYK1 1/20 0.40
HTR6 P50406 1/20 0.40
MGMT P16455 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28000659 0.78 NPC1 (0.47) L3MBTL1NPC1RAB9AMPOTAAR1
SCHEMBL27697197 0.76 CYP19A1 (0.49) RAB9A
SCHEMBL28003702 0.76 NPC1 (0.42) L3MBTL1NPC1RAB9AMPOTAAR1
SCHEMBL28816893 0.76 NPC1 (0.50) L3MBTL1NPC1RAB9AMPOTAAR1
SCHEMBL29520054 0.74 CHRNA7 (0.44) MPO
SCHEMBL29442856 0.74 MAP4K4 (0.45) L3MBTL1NPC1RAB9AMPOTAAR1
SCHEMBL21384071 0.74 MAP4K4 (0.45) L3MBTL1NPC1RAB9AMPOTAAR1
SCHEMBL1774870 0.74 DHFR (0.69)
SCHEMBL3121450 0.73 HTR2C (0.42) L3MBTL1NPC1TAAR1MAOBHTR2C
SCHEMBL15537208 0.72 MAP4K4 (0.60) TLR8TLR7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105189481-A Pyridine cdk9 kinase inhibitors ABBVIE INC 2015-12-23 CN disclosed