SCHEMBL28047870

SCHEMBL28047870

FC(F)(F)c1ccnn1-c1cccnc1

nearest known ligand 0.44

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
CYP11B2 P19099 1/20 0.44
CYP2A6 P11509 4/20 0.42
KDM4E B2RXH2 1/20 0.42
HDAC1 Q13547 1/20 0.41
HDAC6 Q9UBN7 1/20 0.41
CYP3A4 P08684 2/20 0.40
CYP2E1 P05181 2/20 0.38
HTT P42858 1/20 0.38
NTRK1 P04629 1/20 0.37
L3MBTL1 Q9Y468 1/20 0.36
IDO1 P14902 1/20 0.36
TDO2 P48775 1/20 0.36
TRPV1 Q8NER1 1/20 0.36
EP300 Q09472 1/20 0.36
KAT2B Q92831 1/20 0.36
CHRNB2 P17787 1/20 0.36
CHRNA4 P43681 1/20 0.36
NPC1 O15118 1/20 0.36
EPHX2 P34913 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30254265 1.00 CYP11B2 (0.44) CYP11B2CYP2A6KDM4EHDAC1HDAC6
SCHEMBL4988967 0.82 KDM4E (0.56) KDM4ENTRK1
SCHEMBL4886275 0.75 POLB (0.43) KDM4EHTTNTRK1IDO1TDO2
SCHEMBL4883251 0.73 HPGD (0.44) KDM4ENTRK1IDO1TRPV1NPC1
SCHEMBL25417972 0.73 CYP2A6 (0.46) CYP11B2CYP2A6CYP3A4CYP2E1HTT
SCHEMBL2691172 0.73 CYP2A6 (0.49) CYP11B2CYP2A6CYP3A4CYP2E1HTT
SCHEMBL16652179 0.73 POLB (0.66) CYP11B2CYP2A6CYP3A4CYP2E1HTT
SCHEMBL15709954 0.72 CYP11B2 (0.44) CYP11B2CYP2A6CYP3A4CYP2E1HTT
SCHEMBL16927609 0.72 CYP11B2 (0.41) CYP11B2CYP2A6KDM4EHDAC1HDAC6
SCHEMBL4854437 0.71 KDM4E (0.47) KDM4ECYP3A4HTTL3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105324371-A Process for preparing pyridylpyrazole compounds and derivatives thereof from pyridylhydrazine BASF SE 2016-02-10 CN disclosed