SCHEMBL28048822

SCHEMBL28048822

C[Si](C)(C)c1cn(-c2cc[c]cc2)nn1

nearest known ligand 0.44

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
CA12 O43570 1/20 0.44
CA1 P00915 1/20 0.44
CA2 P00918 1/20 0.44
CA9 Q16790 1/20 0.44
NOTUM Q6P988 6/20 0.40
TLR8 Q9NR97 1/20 0.34
FLT3 P36888 4/20 0.34
P2RX7 Q99572 2/20 0.33
MAOA P21397 2/20 0.33
L3MBTL1 Q9Y468 1/20 0.33
RXRA P19793 1/20 0.32
GRIN1 Q05586 1/20 0.32
GRIN2B Q13224 1/20 0.32
MIF P14174 3/20 0.31
CD74 P04233 1/20 0.31
KDM4E B2RXH2 1/20 0.31
MAPT P10636 1/20 0.31
ESRRA P11474 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2886167 0.81 P2RX7 (0.52) CA12CA1CA2CA9NOTUM
SCHEMBL3679115 0.78 CA12 (0.48) CA12CA1CA2CA9NOTUM
SCHEMBL16971964 0.71 NOTUM (0.45) CA12CA1CA2CA9NOTUM
SCHEMBL3753209 0.71 HTT (0.49) CA12CA1CA2CA9MAPT
SCHEMBL15063084 0.70 NOTUM (0.57) CA12CA9NOTUMP2RX7MAOA
SCHEMBL4977179 0.69 BCHE (0.43) CA12CA1CA2CA9NOTUM
SCHEMBL4972496 0.68 BCHE (0.44) CA12CA1CA2CA9NOTUM
SCHEMBL13727128 0.66 RXRA (0.48) CA12CA1CA2CA9RXRA
SCHEMBL24952687 0.65 CA12 (0.46) CA12CA1CA2CA9NOTUM
SCHEMBL2885848 0.64 NOTUM (0.55) CA12CA1CA2CA9NOTUM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105980384-A Macrocyclic compounds having a heterocyclic P2' group as factor XIA inhibitors 百时美施贵宝公司 2016-09-28 CN disclosed
CN-103534253-B Amyloid is had to the compound of affinity NIHON MEDI-PHYSICS CO.,LTD. (JP) 2016-02-24 CN disclosed