SCHEMBL28048853

SCHEMBL28048853

Nc1cc(CCN2CCCC2)c2ccccc2n1

nearest known ligand 0.55

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
NCF1 P14598 5/20 0.55
SLC6A3 Q01959 1/20 0.47
HRH3 Q9Y5N1 4/20 0.47
SIGMAR1 Q99720 1/20 0.46
PARP1 P09874 1/20 0.46
ACP1 P24666 3/20 0.45
SMARCA2 P51531 1/20 0.45
BACE1 P56817 1/20 0.45
HTR2A P28223 1/20 0.44
TOP2A P11388 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28048692 0.87 NCF1 (0.59) NCF1SIGMAR1ACP1TOP2A
SCHEMBL17433848 0.85 NCF1 (0.57) NCF1BACE1
SCHEMBL28825618 0.77 TLR8 (0.56) SLC6A3HRH3SIGMAR1BACE1
SCHEMBL17433976 0.75 NCF1 (0.62) NCF1BACE1
SCHEMBL6665713 0.74 BACE1 (0.53) NCF1BACE1
SCHEMBL6969427 0.74 BACE1 (0.53) NCF1BACE1
SCHEMBL28228172 0.74 HRH3 (0.59) SLC6A3HRH3HTR2A
SCHEMBL4731923 0.72 NCF1 (0.62) NCF1
SCHEMBL17434077 0.72 NCF1 (0.62) NCF1SIGMAR1BACE1
SCHEMBL17433988 0.72 TSHR (0.62) NCF1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105377851-A BET bromodomain inhibitors and therapeutic methods using these inhibitors UNIV MICHIGAN REGENTS 2016-03-02 CN disclosed