SCHEMBL28048974

SCHEMBL28048974

Cc1cc(C)cc(-c2nc(C(=O)O)c(NC(=O)OC(C)(C)C)s2)c1

nearest known ligand 0.43

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
LCK P06239 12/20 0.43
IKBKE Q14164 1/20 0.38
TBK1 Q9UHD2 1/20 0.38
KDM4E B2RXH2 1/20 0.35
GAA P10253 1/20 0.35
RAB9A P51151 1/20 0.35
CYP2C9 P11712 1/20 0.34
CYP2C19 P33261 1/20 0.34
NPSR1 Q6W5P4 1/20 0.34
RAF1 P04049 1/20 0.34
BRD9 Q9H8M2 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2521682 0.85 KDM4E (0.48) LCKTBK1KDM4EGAARAB9A
SCHEMBL15573656 0.85 LCK (0.41) LCKCYP2C9CYP2C19NPSR1
SCHEMBL2524367 0.82 KDM4E (0.48) LCKKDM4EGAARAB9ACYP2C9
SCHEMBL2520688 0.81 USP30 (0.40) LCKKDM4EGAA
SCHEMBL2520080 0.81 KMT2A (0.45) LCKKDM4ERAB9A
SCHEMBL29019243 0.80 LCK (0.39) LCKBRD9
SCHEMBL27866744 0.80 ALDH1A1 (0.46) KDM4ERAB9A
SCHEMBL19912149 0.80 HDAC6 (0.37) LCKKDM4ERAB9ANPSR1BRD9
SCHEMBL14800615 0.80 PIM1 (0.37) LCK
SCHEMBL6523055 0.80 LCK (0.47) LCKGAARAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-102625807-B 4-Substituted pyridin-3-yl-carboxamide compounds and methods of use HOFFMAN-LA ROCHE LTD. (CH) 2016-03-09 CN disclosed