SCHEMBL28049495

SCHEMBL28049495

COc1cc(N(c2ccc(F)c(Cl)c2)c2cc(N)ncn2)ccc1N

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDR P35968 3/20 0.40
EGFR P00533 10/20 0.37
AURKA O14965 1/20 0.37
ERBB2 P04626 1/20 0.37
INSR P06213 1/20 0.37
FBP1 P09467 1/20 0.37
PDGFRB P09619 1/20 0.37
FLT4 P35916 1/20 0.37
CLK1 P49759 1/20 0.37
EPHB4 P54760 1/20 0.37
TEK Q02763 1/20 0.37
AURKB Q96GD4 1/20 0.37
LTC4S Q16873 1/20 0.36
FYN P06241 1/20 0.35
CSF1R P07333 2/20 0.35
ALDH1A1 P00352 2/20 0.35
CYP3A4 P08684 2/20 0.35
KIT P10721 1/20 0.34
DYRK1A Q13627 1/20 0.34
GRM1 Q13255 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL691612 0.84 KDR (0.38) KDREGFRAURKAERBB2INSR
SCHEMBL690517 0.75 MAPK1 (0.36) EGFRAURKAGRM1
SCHEMBL690859 0.75 EGFR (0.37) KDREGFRERBB2ALDH1A1CYP3A4
SCHEMBL690928 0.72 CYP3A4 (0.36) EGFRALDH1A1CYP3A4TSHRTDP1
SCHEMBL28056977 0.71 EGFR (0.55) KDREGFRAURKAERBB2INSR
SCHEMBL25142 0.68 EGFR (0.51) KDREGFRAURKAERBB2INSR
SCHEMBL654423 0.65 MAPK1 (0.42) EPHB4ALDH1A1
SCHEMBL14495631 0.64 ALDH1A1 (0.53) ALDH1A1CYP3A4TSHRHSD17B10TDP1
SCHEMBL15877055 0.63 KIT (0.67) KDREGFRAURKAERBB2INSR
SCHEMBL4805640 0.62 ADORA2A (0.46) ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-101902911-B Heteroaryl compounds and uses thereof AVILA THERAPEUTICS, INC. (US) 2015-12-16 CN disclosed