SCHEMBL28050770

SCHEMBL28050770

[c]1cccc(COc2ccc3c(c2)CCCC3)c1

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 5/20 0.53
RAB9A P51151 5/20 0.53
RXRB P28702 4/20 0.53
RXRA P19793 3/20 0.53
RXRG P48443 3/20 0.53
POLB P06746 1/20 0.53
GFER P55789 1/20 0.53
PAX8 Q06710 1/20 0.53
KLF5 Q13887 1/20 0.53
MRGPRX4 Q96LA9 1/20 0.53
L3MBTL1 Q9Y468 1/20 0.53
HRH3 Q9Y5N1 9/20 0.52
SMN1; SMN2 Q16637 3/20 0.50
ALDH1A1 P00352 1/20 0.50
TP53 P04637 1/20 0.50
MAPT P10636 1/20 0.50
LMNA P02545 1/20 0.50
GAA P10253 1/20 0.50
HPGD P15428 1/20 0.50
CYP2D6 P10635 2/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30299191 0.83 HRH3 (0.72) NPC1RAB9ARXRBRXRARXRG
SCHEMBL921884 0.80 HRH3 (0.43) NPC1RAB9ARXRBRXRARXRG
SCHEMBL12472442 0.80 HRH3 (0.72) NPC1RAB9ARXRBRXRARXRG
SCHEMBL920751 0.77 HRH3 (0.43) NPC1RAB9ARXRBRXRARXRG
SCHEMBL919605 0.74 MAOB (0.50) NPC1RAB9AL3MBTL1SMN1; SMN2MAPT
SCHEMBL8462058 0.74 RXRB (0.61) NPC1RAB9ARXRBRXRARXRG
SCHEMBL11961605 0.73 NPC1 (0.64) NPC1RAB9ARXRBRXRARXRG
SCHEMBL6507309 0.73 MAOB (0.50) ALDH1A1MAOB
SCHEMBL2264253 0.73 MAOB (0.56) HRH3MAOAMAOBKDM4E
SCHEMBL30714042 0.72 ADRA1D (0.60) NPC1RAB9ARXRBRXRARXRG

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105175360-B Ether-type aryl bridged piperazine derivatives and its salt, preparation method and purposes 洛阳师范学院 2017-12-15 CN disclosed
CN-105175360-A Ether aryl piperazine derivatives, and salts, preparation methods and application thereof UNIV LUOYANG NORMAL 2015-12-23 CN disclosed