SCHEMBL28051973

SCHEMBL28051973

Cc1ccc(-c2ccnc(C(N)=O)c2)cn1

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GSK3B P49841 3/20 0.52
PIK3CB P42338 2/20 0.51
MKNK1 Q9BUB5 2/20 0.46
MKNK2 Q9HBH9 2/20 0.46
CCNC P24863 2/20 0.46
CDK8 P49336 2/20 0.46
CYP11B2 P19099 1/20 0.43
KCNH2 Q12809 1/20 0.43
ATM Q13315 1/20 0.43
ATR Q13535 1/20 0.43
PIK3CD O00329 1/20 0.42
PIK3CA P42336 1/20 0.42
PI4KA P42356 1/20 0.42
PIK3CG P48736 1/20 0.42
PI4KB Q9UBF8 1/20 0.42
GABRA1 P14867 2/20 0.42
TLR8 Q9NR97 1/20 0.41
TLR7 Q9NYK1 1/20 0.41
ADORA3 P0DMS8 1/20 0.41
TSHR P16473 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29859342 0.85 KMO (0.57) GSK3BPIK3CBPIK3CDPIK3CAPI4KA
SCHEMBL945743 0.85 GSK3B (0.63) GSK3BPIK3CBMKNK1MKNK2TLR8
SCHEMBL27772527 0.81 MKNK1 (0.51) GSK3BPIK3CBMKNK1MKNK2CCNC
Hydrochloric Acid SCHEMBL9792812 0.80 MKNK1 (0.52) GSK3BPIK3CBMKNK1MKNK2CCNC
SCHEMBL956760 0.79 GSK3B (0.45) GSK3BPIK3CBMKNK1MKNK2KCNH2
SCHEMBL933914 0.79 MKNK1 (0.59) MKNK1MKNK2CYP11B2ADORA3TSHR
SCHEMBL30761107 0.79 MKNK1 (0.59) MKNK1MKNK2CYP11B2ADORA3TSHR
SCHEMBL3346810 0.77 MKNK1 (0.52) PIK3CBMKNK1MKNK2CYP11B2KCNH2
SCHEMBL3422269 0.77 DYRK1A (0.56) PIK3CBPIK3CDPIK3CAPI4KAPIK3CG
SCHEMBL12269997 0.76 CCNT1 (0.55) GSK3BMKNK1MKNK2CCNCCDK8

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105658639-A Alkynyl alcohols and methods of use 豪夫迈·罗氏有限公司 2016-06-08 CN disclosed