SCHEMBL956760

SCHEMBL956760

CC(C)(O)c1ccc(-c2ccnc(C(N)=O)c2)cn1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GSK3B P49841 1/20 0.45
SYK P43405 7/20 0.42
PIK3CB P42338 1/20 0.41
CCR7 P32248 1/20 0.41
CCR6 P51684 1/20 0.41
ADORA3 P0DMS8 1/20 0.40
TSHR P16473 1/20 0.40
MC4R P32245 1/20 0.40
ADRA1A P35348 1/20 0.40
MC3R P41968 1/20 0.40
MKNK1 Q9BUB5 1/20 0.40
MKNK2 Q9HBH9 1/20 0.40
MYC P01106 1/20 0.40
KCNH2 Q12809 1/20 0.39
PDE4A P27815 1/20 0.38
PDE4B Q07343 1/20 0.38
PDE4C Q08493 1/20 0.38
PDE4D Q08499 1/20 0.38
HDAC1 Q13547 1/20 0.37
KMO O15229 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL946562 0.87 KMO (0.51) SYKKCNH2HDAC1KMO
Hydrochloric Acid SCHEMBL934035 0.86 KMO (0.50) SYKKCNH2HDAC1KMO
SCHEMBL934021 0.80 SYK (0.41) SYKKCNH2
SCHEMBL945743 0.80 GSK3B (0.63) GSK3BPIK3CBADORA3TSHRMC4R
SCHEMBL28051973 0.79 GSK3B (0.52) GSK3BPIK3CBADORA3TSHRMC4R
SCHEMBL944085 0.79 CCNT1 (0.50) GSK3BSYKCCR6
Hydrochloric Acid SCHEMBL9792812 0.76 MKNK1 (0.52) GSK3BPIK3CBADORA3TSHRMC4R
SCHEMBL943650 0.75 LRRK2 (0.51) CCR7CCR6MKNK1MKNK2MYC
SCHEMBL27772527 0.73 MKNK1 (0.51) GSK3BPIK3CBMKNK1MKNK2MYC
SCHEMBL30595907 0.73 OPRM1 (0.42) GSK3BADORA3TSHRMC4RADRA1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011008709-A1 APOPTOSIS SIGNAL-REGULATING KINASE INHIBITORS GILEAD SCIENCES, INC. (US) 2011-01-20 WO claimed