SCHEMBL28052184

SCHEMBL28052184

COc1ccc(Cc2nc(N)nc3nc(C=O)[nH]c23)cc1OC

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 1/20 0.44
DHFR P00374 1/20 0.43
HTT P42858 1/20 0.43
CA2 P00918 1/20 0.41
ALDH1A1 P00352 4/20 0.41
CYP3A4 P08684 3/20 0.41
LMNA P02545 3/20 0.41
CYP2C9 P11712 2/20 0.41
TSHR P16473 2/20 0.41
CYP2C19 P33261 2/20 0.41
USP2 O75604 2/20 0.41
MAPK1 P28482 2/20 0.41
SMN1; SMN2 Q16637 2/20 0.41
HIF1A Q16665 2/20 0.41
PDE10A Q9Y233 2/20 0.41
PDE2A O00408 1/20 0.41
ABCC4 O15439 1/20 0.41
PDE5A O76074 1/20 0.41
ABCB11 O95342 1/20 0.41
CYP1A2 P05177 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1855271 0.73 DHFR (0.53) DHFRHTTALDH1A1HPGDPOLB
SCHEMBL30647980 0.67 DHFR (0.48) DHFRHTTCA2ALDH1A1CYP3A4
SCHEMBL11831045 0.65 DHFR (0.58) DHFRHTTCA2ALDH1A1CYP2D6
SCHEMBL1859068 0.64 HSP90AA1 (0.69) KMT2ADHFRHTTCA2ALDH1A1
SCHEMBL9828253 0.64 CA2 (0.77) DHFRHTTCA2ALDH1A1CYP3A4
SCHEMBL1053909 0.64 DHFR (0.50) DHFRHTTCA2
SCHEMBL11006578 0.64 DHFR (0.71) DHFRHTT
SCHEMBL1855267 0.64 DHFR (0.53) KMT2ADHFRHTTCA2ALDH1A1
SCHEMBL2095593 0.63 CA2 (1.00) CA2ALDH1A1CYP3A4LMNACYP2C9
SCHEMBL11567021 0.63 DHFR (0.67) DHFRHTTCA2ALDH1A1HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-103261202-B As the fused tricyclic compounds of adenosine receptor antagonists ADVINUS THERAPEUTICS LTD. (IN) 2016-01-20 CN disclosed