SCHEMBL28052676

SCHEMBL28052676

NC(=O)c1cccc(-c2ccncc2)n1

nearest known ligand 0.57

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SCN9A Q15858 10/20 0.57
IRAK4 Q9NWZ3 1/20 0.54
MAP2K3 P46734 3/20 0.54
DGAT1 O75907 1/20 0.50
MAPK14 Q16539 1/20 0.49
CDC7 O00311 1/20 0.44
CCNE1 P24864 1/20 0.44
CDK2 P24941 1/20 0.44
DBF4 Q9UBU7 1/20 0.44
CASP1 P29466 1/20 0.44
PLK4 O00444 1/20 0.43
MAPK13 O15264 1/20 0.43
DYRK3 O43781 1/20 0.43
ROCK2 O75116 1/20 0.43
RPS6KA5 O75582 1/20 0.43
PRKD3 O94806 1/20 0.43
MAP4K4 O95819 1/20 0.43
CHEK2 O96017 1/20 0.43
PIM1 P11309 1/20 0.43
PHKG2 P15735 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29911672 1.00 SCN9A (0.57) SCN9AIRAK4MAP2K3DGAT1MAPK14
SCHEMBL29648185 0.85 DGAT1 (0.56) SCN9AIRAK4MAP2K3DGAT1CASP1
SCHEMBL608430 0.85 DGAT1 (0.56) SCN9AIRAK4MAP2K3DGAT1CASP1
SCHEMBL1944293 0.84 KDM4E (0.57) SCN9AIRAK4MAP2K3CDC7DBF4
SCHEMBL28324757 0.83 SCN9A (0.59) SCN9AIRAK4PKN1PKN2MKNK2
SCHEMBL29505512 0.83 SCN9A (0.59) SCN9AIRAK4PKN1PKN2MKNK2
SCHEMBL9792961 0.82 PIM1 (0.50) SCN9AIRAK4DGAT1PIM1
SCHEMBL16129931 0.82 SCN9A (0.56) SCN9AIRAK4MAP2K3DGAT1
SCHEMBL16129942 0.82 ALDH1A1 (0.62) SCN9AIRAK4DGAT1PIM1
Hydrochloric Acid SCHEMBL29855542 0.81 SCN9A (0.58) SCN9AIRAK4PKN1PKN2MKNK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-103282360-B CXCR4 receptor antagonist PROXIMAGEN LTD. (GB) 2016-03-30 CN disclosed