SCHEMBL28053003

SCHEMBL28053003

O=C(O)NCCC(O)c1cccc(C#CC2CCCC2)c1

nearest known ligand 0.42

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
PTGES O14684 3/20 0.42
HAO1 Q9UJM8 5/20 0.40
FFAR1 O14842 2/20 0.40
FFAR4 Q5NUL3 2/20 0.40
GRM5 P41594 1/20 0.36
EPHX2 P34913 2/20 0.36
ALOX5 P09917 1/20 0.36
KDM4E B2RXH2 1/20 0.35
MTNR1A P48039 1/20 0.35
MTNR1B P49286 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16032074 0.90 HAO1 (0.43) PTGESHAO1FFAR1GRM5EPHX2
SCHEMBL237114 0.86 PTGES (0.37) PTGESHAO1FFAR1FFAR4EPHX2
SCHEMBL3837431 0.85 SLC6A3 (0.34) PTGESGRM5EPHX2ALOX5KDM4E
SCHEMBL237238 0.84 DDB1 (0.40) PTGESHAO1GRM5
SCHEMBL234717 0.84 EPHX1 (0.39) PTGESHAO1FFAR1FFAR4GRM5
SCHEMBL236453 0.84 EPHX1 (0.39) PTGESHAO1FFAR1FFAR4GRM5
SCHEMBL233588 0.83 HAO1 (0.37) PTGESHAO1FFAR1FFAR4
SCHEMBL3839542 0.83 PTPN11 (0.41) PTGESFFAR1GRM5EPHX2ALOX5
SCHEMBL236160 0.82 PTGES (0.39) PTGESHAO1FFAR1GRM5EPHX2
SCHEMBL233144 0.82 HAO1 (0.38) PTGESHAO1FFAR1FFAR4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105541769-A Alkynyl phenyl derivative compounds for treating ophthalmic diseases and disorders ACUCELA INC 2016-05-04 CN disclosed
CN-103664637-B Be used for the treatment of ophthalmic diseases and disorderly alkynyl phenyl derivative compounds ACUCELA INC. (US) 2016-02-03 CN disclosed