SCHEMBL28053317

SCHEMBL28053317

O=C(O)c1ccc2c(n1)-c1ccccc1CC2

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 6/20 0.51
ALDH1A1 P00352 4/20 0.51
CYP1A2 P05177 3/20 0.49
CYP3A4 P08684 3/20 0.49
CYP2C19 P33261 2/20 0.49
GAA P10253 1/20 0.49
GSR P00390 1/20 0.47
SRD5A1 P18405 1/20 0.46
SRD5A2 P31213 1/20 0.46
PTGER1 P34995 1/20 0.45
POLB P06746 2/20 0.45
LMNA P02545 2/20 0.44
MGAM O43451 1/20 0.43
HPGD P15428 1/20 0.43
NOTUM Q6P988 1/20 0.43
ALOX15 P16050 1/20 0.42
TSHR P16473 1/20 0.42
ACMSD Q8TDX5 1/20 0.42
TDP1 Q9NUW8 1/20 0.42
CYP2D6 P10635 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28600177 0.72 NPY5R (0.49) KDM4EALDH1A1CYP1A2CYP3A4CYP2C19
SCHEMBL14610321 0.72 KDM4E (0.48) KDM4EALDH1A1SRD5A2LMNAMGAM
Hydrochloric Acid SCHEMBL9544492 0.72 BCHE (0.42) KDM4EALDH1A1CYP1A2CYP3A4CYP2C19
SCHEMBL29365290 0.72 KDM4E (0.50) KDM4EALDH1A1CYP1A2CYP3A4CYP2C19
SCHEMBL6766148 0.71 ALDH1A1 (0.41) KDM4EALDH1A1LMNAMGAMHPGD
SCHEMBL9544495 0.70 DRD4 (0.41) KDM4EALDH1A1CYP1A2CYP3A4CYP2C19
SCHEMBL2837730 0.68 KDM4E (0.54) KDM4EALDH1A1CYP3A4GAAPOLB
SCHEMBL8172786 0.68 KDM4E (1.00) KDM4EALDH1A1GSRPOLBHPGD
SCHEMBL319496 0.68 MGAM (0.44) KDM4EMGAMALOX15TSHRACMSD
SCHEMBL11794463 0.68 ALDH1A1 (0.52) KDM4EALDH1A1CYP1A2CYP2C19GAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105294678-A 9-fluoro-6,7-dihydro-8-(4-hydroxy-1-piperidinyl)-5-methyl-1-oxo-1H, 5H-benzo-quinoline-2-carboxylic acid preparation method NANJING GRITPHARMA CO LTD 2016-02-03 CN disclosed
CN-105294678-A 9-fluoro-6,7-dihydro-8-(4-hydroxy-1-piperidinyl)-5-methyl-1-oxo-1H, 5H-benzo-quinoline-2-carboxylic acid preparation method NANJING GRITPHARMA CO LTD 2016-02-03 CN disclosed