SCHEMBL28053335

SCHEMBL28053335

COc1cnc(Cl)nc1-c1ccc(S(N)(=O)=O)cc1-c1nc(Cl)ncc1OC

nearest known ligand 0.42

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
CA2 P00918 6/20 0.42
CA9 Q16790 6/20 0.42
CA12 O43570 5/20 0.42
CA1 P00915 5/20 0.42
PTGS1 P23219 5/20 0.41
PTGS2 P35354 5/20 0.41
EGFR P00533 1/20 0.41
KDR P35968 1/20 0.41
GAA P10253 2/20 0.41
PDK1 Q15118 1/20 0.39
TDP2 O95551 1/20 0.39
NSD2 O96028 1/20 0.39
HK1 P19367 1/20 0.39
PAX8 Q06710 1/20 0.39
IKBKB O14920 1/20 0.39
CA4 P22748 1/20 0.39
POLB P06746 1/20 0.38
PKM P14618 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28053355 0.80 KDM4E (0.41) CA2CA9CA12CA1PTGS1
SCHEMBL2315314 0.68 PTGS2 (0.66) CA2CA9CA12CA1PTGS1
SCHEMBL30540198 0.68 CA2 (0.40) CA2CA9CA12CA1GAA
SCHEMBL29057759 0.68 CA2 (0.40) CA2CA9CA12CA1GAA
SCHEMBL24478222 0.66 MAPT (0.67) CA2CA9CA12CA1PTGS1
SCHEMBL30823485 0.66 MAPT (0.67) CA2CA9CA12CA1PTGS1
SCHEMBL1808957 0.66 PTGS2 (0.69) CA2CA9CA12CA1PTGS1
SCHEMBL30269805 0.66 PTGS2 (0.52) CA2CA9CA12CA1PTGS1
SCHEMBL11335088 0.65 PTGS2 (0.42) CA2CA9CA12CA1PTGS1
SCHEMBL25551994 0.65 KMT2A (0.50) GAAPDK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105377837-B N (heteroaryl) sulfamide derivative as S100 inhibitor 活跃生物技术有限公司 2017-08-04 CN disclosed
CN-105377837-A N-(heteroaryl)-sulfonamide derivatives useful as S100-inhibitors ACTIVE BIOTECH AB 2016-03-02 CN disclosed