SCHEMBL28053556

SCHEMBL28053556

CC(=O)Oc1ccnc(C2CC2)c1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LMNA P02545 2/20 0.41
CYP3A4 P08684 1/20 0.41
HDAC4 P56524 4/20 0.41
HDAC3 O15379 1/20 0.41
HDAC7 Q8WUI4 1/20 0.41
HDAC8 Q9BY41 1/20 0.41
HDAC6 Q9UBN7 1/20 0.41
HDAC9 Q9UKV0 1/20 0.41
HDAC5 Q9UQL6 1/20 0.41
KMT2A Q03164 1/20 0.39
KDM4E B2RXH2 3/20 0.38
ACHE P22303 2/20 0.38
PROKR1 Q8TCW9 1/20 0.37
ALDH1A1 P00352 1/20 0.37
F2 P00734 1/20 0.37
GLA P06280 1/20 0.37
HPGD P15428 1/20 0.37
SMN1; SMN2 Q16637 1/20 0.37
MAPT P10636 1/20 0.36
HSD17B10 Q99714 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15880899 0.84 MEN1 (0.46) HDAC4HDAC3HDAC7HDAC8HDAC6
SCHEMBL17669635 0.79 CCR1 (0.55) LMNACYP3A4KMT2AKDM4EACHE
SCHEMBL30943495 0.78 CCR1 (0.59) CYP3A4HDAC4HDAC3HDAC7HDAC8
SCHEMBL7856828 0.78 CCR1 (0.59) CYP3A4HDAC4HDAC3HDAC7HDAC8
SCHEMBL25984345 0.75 PROKR1 (0.48) HDAC4HDAC3HDAC7HDAC8HDAC6
SCHEMBL28025233 0.74 HDAC4 (0.39) LMNACYP3A4HDAC4KMT2AKDM4E
SCHEMBL9670309 0.74 LMNA (0.47) LMNACYP3A4KMT2AKDM4EACHE
SCHEMBL7674985 0.74 LMNA (0.52) LMNACYP3A4KDM4EACHEALDH1A1
SCHEMBL25348842 0.73 LMNA (0.46) LMNACYP3A4KMT2AKDM4EACHE
Hydrochloric Acid SCHEMBL10529996 0.73 LMNA (0.50) LMNACYP3A4KDM4EACHEALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105452233-A Piperidine and azepane derivatives as prokineticin receptor modulators TAKEDA PHARMACEUTICALS CO 2016-03-30 CN disclosed