SCHEMBL28053852

SCHEMBL28053852

C=CC(=O)Nc1ccc(OC)c(Nc2nccc(Nc3ccc(N4CCN(C)CC4)cc3OC)n2)c1

nearest known ligand 0.78

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
EGFR P00533 13/20 0.78
JAK3 P52333 4/20 0.74
CTSC P53634 4/20 0.64
FLT3 P36888 2/20 0.62
BLK P51451 2/20 0.62
ALK Q9UM73 2/20 0.62
PLK4 O00444 1/20 0.61
GAK O14976 1/20 0.61
NUAK1 O60285 1/20 0.61
JAK2 O60674 1/20 0.61
BMX P51813 1/20 0.61
PTK2 Q05397 1/20 0.61
BTK Q06187 1/20 0.61
ITK Q08881 1/20 0.61
ERBB4 Q15303 1/20 0.61
DCLK3 Q9C098 1/20 0.61
NUAK2 Q9H093 1/20 0.61
EML4 Q9HC35 1/20 0.61
EIF2AK4 Q9P2K8 1/20 0.61

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28452560 0.96 EGFR (0.73) EGFRJAK3CTSCFLT3BLK
SCHEMBL28053996 0.92 ALK (0.75) EGFRJAK3ALKGAKPTK2
SCHEMBL28447722 0.91 EGFR (0.78) EGFRJAK3ALK
SCHEMBL28053986 0.91 EGFR (0.80) EGFRJAK3CTSCFLT3BLK
SCHEMBL28053999 0.90 EGFR (0.65) EGFRJAK3CTSCFLT3BLK
SCHEMBL17059644 0.88 EGFR (1.00) EGFRJAK3CTSCFLT3BLK
SCHEMBL28053891 0.87 JAK3 (0.77) EGFRJAK3CTSCFLT3BLK
SCHEMBL17209827 0.85 JAK3 (1.00) EGFRJAK3FLT3BLKJAK2
SCHEMBL28053991 0.84 JAK3 (0.73) EGFRJAK3CTSCFLT3BLK
SCHEMBL28915867 0.83 EGFR (0.75) EGFRJAK3ALKGAKPTK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105384694-B Substituted aminopyrimidine derivative and preparation method and pharmaceutical application thereof 四川海思科制药有限公司 2020-09-04 CN disclosed
CN-105384694-A Substituted aminopyrimidine derivative, preparation method therefor and pharmaceutical application thereof SICHUAN HAISCO PHARMACEUTICAL CO LTD 2016-03-09 CN disclosed