SCHEMBL28053891

SCHEMBL28053891

C=CC(=O)Nc1ccc(OC)c(Nc2ncc(Cl)c(Nc3ccc(N4CCN(C)CC4)cc3OC)n2)c1

nearest known ligand 0.77

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
JAK3 P52333 9/20 0.77
EGFR P00533 9/20 0.76
FLT3 P36888 3/20 0.74
BLK P51451 3/20 0.74
JAK2 O60674 2/20 0.74
BTK Q06187 2/20 0.74
ITK Q08881 2/20 0.74
JAK1 P23458 1/20 0.74
TTK P33981 1/20 0.74
TXK P42681 1/20 0.74
PLK4 O00444 1/20 0.73
GAK O14976 1/20 0.73
NUAK1 O60285 1/20 0.73
BMX P51813 1/20 0.73
CTSC P53634 1/20 0.73
PTK2 Q05397 1/20 0.73
ERBB4 Q15303 1/20 0.73
DCLK3 Q9C098 1/20 0.73
NUAK2 Q9H093 1/20 0.73
EML4 Q9HC35 1/20 0.73

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28053991 0.97 JAK3 (0.73) JAK3EGFRFLT3BLKJAK2
SCHEMBL28579656 0.92 EGFR (0.83) EGFRALKMAPK3
SCHEMBL28053865 0.92 EGFR (0.83) JAK3EGFRFLT3JAK2BTK
Hydrochloric Acid SCHEMBL28053870 0.91 EGFR (0.82) JAK3EGFRFLT3JAK2BTK
SCHEMBL10128042 0.91 EGFR (0.86) JAK3EGFRFLT3BLKJAK2
SCHEMBL28589279 0.89 ALK (0.71) JAK3EGFRBTKEML4ALK
SCHEMBL17209776 0.87 JAK3 (1.00) JAK3EGFRFLT3BLKJAK2
SCHEMBL28053852 0.87 EGFR (0.78) JAK3EGFRFLT3BLKJAK2
SCHEMBL10155134 0.86 EGFR (1.00) JAK3EGFRFLT3BLKJAK2
SCHEMBL28595246 0.86 MAPK3 (0.81) EGFRALKMAPK3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105384694-B Substituted aminopyrimidine derivative and preparation method and pharmaceutical application thereof 四川海思科制药有限公司 2020-09-04 CN disclosed
CN-105384694-A Substituted aminopyrimidine derivative, preparation method therefor and pharmaceutical application thereof SICHUAN HAISCO PHARMACEUTICAL CO LTD 2016-03-09 CN disclosed